Compile Data Set for Download or QSAR
Report error Found 240 Enz. Inhib. hit(s) with all data for entry = 11517
TargetLIM domain kinase 2(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622419BDBM622419(US20230312576, Compound 75)
Affinity DataKi:  2.73nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622459BDBM622459(US20230312576, Compound 136)
Affinity DataKi:  2.75nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 2(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622485BDBM622485(US20230312576, Compound 198)
Affinity DataKi:  2.89nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 2(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622495BDBM622495(US20230312576, Compound 222)
Affinity DataKi:  2.96nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622485BDBM622485(US20230312576, Compound 198)
Affinity DataKi:  3.08nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622431BDBM622431(US20230312576, Compound 93)
Affinity DataKi:  3.71nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 2(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622445BDBM622445(US20230312576, Compound 122)
Affinity DataKi:  4.02nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622495BDBM622495(US20230312576, Compound 222)
Affinity DataKi:  4.59nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 2(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622421BDBM622421(US20230312576, Compound 77)
Affinity DataKi:  4.64nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622493BDBM622493(US20230312576, Compound 216)
Affinity DataKi:  4.88nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622494BDBM622494(US20230312576, Compound 219)
Affinity DataKi:  4.93nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622460BDBM622460(US20230312576, Compound 137)
Affinity DataKi:  4.97nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622433BDBM622433(US20230312576, Compound 110)
Affinity DataKi:  5nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622438BDBM622438(US20230312576, Compound 115)
Affinity DataKi:  5.37nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 2(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622494BDBM622494(US20230312576, Compound 219)
Affinity DataKi:  5.46nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622434BDBM622434(US20230312576, Compound 111)
Affinity DataKi:  5.78nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622444BDBM622444(US20230312576, Compound 121)
Affinity DataKi:  6.10nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622447BDBM622447(US20230312576, Compound 124)
Affinity DataKi:  6.49nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622427BDBM622427(US20230312576, Compound 89)
Affinity DataKi:  6.60nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 2(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622420BDBM622420(US20230312576, Compound 76)
Affinity DataKi:  6.95nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622435BDBM622435(US20230312576, Compound 112)
Affinity DataKi:  7nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622445BDBM622445(US20230312576, Compound 122)
Affinity DataKi:  7.11nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622436BDBM622436(US20230312576, Compound 113)
Affinity DataKi:  7.13nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 2(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622490BDBM622490(US20230312576, Compound 208)
Affinity DataKi:  7.57nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622442BDBM622442(US20230312576, Compound 119)
Affinity DataKi:  7.98nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 2(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622398BDBM622398(US20230312576, Compound 30)
Affinity DataKi:  8.15nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622450BDBM622450(US20230312576, Compound 127)
Affinity DataKi:  8.19nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 2(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622410BDBM622410(US20230312576, Compound 63 | US20230312576, Compou...)
Affinity DataKi:  8.49nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 2(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622414BDBM622414(US20230312576, Compound 66)
Affinity DataKi:  8.49nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 2(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622460BDBM622460(US20230312576, Compound 137)
Affinity DataKi:  8.59nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 2(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622454BDBM622454(US20230312576, Compound 131)
Affinity DataKi:  8.73nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 2(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622408BDBM622408(US20230312576, Compound 49a-49b)
Affinity DataKi:  8.89nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622430BDBM622430(US20230312576, Compound 92)
Affinity DataKi:  8.99nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 2(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622470BDBM622470(US20230312576, Compound 175)
Affinity DataKi:  9.66nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 2(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622418BDBM622418(US20230312576, Compound 74)
Affinity DataKi:  9.67nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 2(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622486BDBM622486(US20230312576, Compound 200)
Affinity DataKi:  9.83nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 2(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622424BDBM622424(US20230312576, Compound 81)
Affinity DataKi:  9.98nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622437BDBM622437(US20230312576, Compound 114)
Affinity DataKi:  9.98nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622404BDBM622404(US20230312576, Compound 40)
Affinity DataKi:  10.6nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622408BDBM622408(US20230312576, Compound 49a-49b)
Affinity DataKi:  10.8nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 2(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622423BDBM622423(US20230312576, Compound 79)
Affinity DataKi:  10.9nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622446BDBM622446(US20230312576, Compound 123)
Affinity DataKi:  11.5nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 2(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622393BDBM622393(US20230312576, Compound 22)
Affinity DataKi:  11.9nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622470BDBM622470(US20230312576, Compound 175)
Affinity DataKi:  12nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622399BDBM622399(US20230312576, Compound 31)
Affinity DataKi:  12.4nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622492BDBM622492(US20230312576, Compound 213)
Affinity DataKi:  12.9nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622388BDBM622388(US20230312576, Compound 17)
Affinity DataKi:  13.2nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 1(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622424BDBM622424(US20230312576, Compound 81)
Affinity DataKi:  13.3nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 2(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622404BDBM622404(US20230312576, Compound 40)
Affinity DataKi:  13.4nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

TargetLIM domain kinase 2(Human)
Centre National De La Recherche Scientifique

US Patent
LigandChemical structure of BindingDB Monomer ID 622397BDBM622397(US20230312576, Compound 29)
Affinity DataKi:  13.7nMAssay Description:Inhibition of LIMK1 and LIMK2. Inhibition of LIMK1 and LIMK2 was measured with Lanthascreen Eu binding assay (Life Technologies). This TR-FRET assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
US Patent

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