Compile Data Set for Download or QSAR
Report error Found 103 Enz. Inhib. hit(s) with all data for entry = 6107
TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109106BDBM109106(US8609852, 13)
Affinity DataKi:  0.600nM ΔG°:  -52.6kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109136BDBM109136(US8609852, 43)
Affinity DataKi:  0.650nM ΔG°:  -52.4kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109101BDBM109101(US8609852, 7)
Affinity DataKi:  0.700nM ΔG°:  -52.3kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109157BDBM109157(US8609852, 64)
Affinity DataKi:  0.800nM ΔG°:  -51.9kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109121BDBM109121(US8609852, 28)
Affinity DataKi:  0.900nM ΔG°:  -51.6kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109102BDBM109102(US8609852, 8)
Affinity DataKi:  0.900nM ΔG°:  -51.6kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109115BDBM109115(US8609852, 117 | US8609852, 34)
Affinity DataKi:  0.900nM ΔG°:  -51.6kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109120BDBM109120(US8609852, 27)
Affinity DataKi:  1nM ΔG°:  -51.4kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109176BDBM109176(US8609852, 85)
Affinity DataKi:  1nM ΔG°:  -51.4kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109182BDBM109182(US8609852, 91)
Affinity DataKi:  1nM ΔG°:  -51.4kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109099BDBM109099(US8609852, 5)
Affinity DataKi:  1nM ΔG°:  -51.4kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109115BDBM109115(US8609852, 117 | US8609852, 34)
Affinity DataKi:  1nM ΔG°:  -51.4kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109105BDBM109105(US8609852, 12)
Affinity DataKi:  1.10nM ΔG°:  -51.1kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109100BDBM109100(US8609852, 6)
Affinity DataKi:  1.20nM ΔG°:  -50.9kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 50181753BDBM50181753(US8609852, 78 | CHEMBL202307 | 3-[(2-methyl-4-thia...)
Affinity DataKi:  1.40nM ΔG°:  -50.5kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109113BDBM109113(US8609852, 20)
Affinity DataKi:  1.40nM ΔG°:  -50.5kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109153BDBM109153(US8609852, 60)
Affinity DataKi:  1.5nM ΔG°:  -50.4kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109147BDBM109147(US8609852, 54)
Affinity DataKi:  1.5nM ΔG°:  -50.4kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109114BDBM109114(US8609852, 21)
Affinity DataKi:  1.5nM ΔG°:  -50.4kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109151BDBM109151(US8609852, 58)
Affinity DataKi:  1.5nM ΔG°:  -50.4kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109194BDBM109194(US8609852, 103)
Affinity DataKi:  1.60nM ΔG°:  -50.2kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109116BDBM109116(US8609852, 23)
Affinity DataKi:  1.60nM ΔG°:  -50.2kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109139BDBM109139(US8609852, 46)
Affinity DataKi:  2nM ΔG°:  -49.7kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109137BDBM109137(US8609852, 44)
Affinity DataKi:  2nM ΔG°:  -49.7kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109173BDBM109173(US8609852, 82)
Affinity DataKi:  2nM ΔG°:  -49.7kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109096BDBM109096(US8609852, 2)
Affinity DataKi:  2nM ΔG°:  -49.7kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109145BDBM109145(US8609852, 52)
Affinity DataKi:  2nM ΔG°:  -49.7kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109119BDBM109119(US8609852, 26)
Affinity DataKi:  2nM ΔG°:  -49.7kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109166BDBM109166(US8609852, 73)
Affinity DataKi:  2nM ΔG°:  -49.7kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109180BDBM109180(US8609852, 89)
Affinity DataKi:  2nM ΔG°:  -49.7kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109123BDBM109123(US8609852, 30)
Affinity DataKi:  2.30nM ΔG°:  -49.3kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109108BDBM109108(US8609852, 15)
Affinity DataKi:  2.60nM ΔG°:  -49.0kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109117BDBM109117(US8609852, 24)
Affinity DataKi:  2.60nM ΔG°:  -49.0kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109098BDBM109098(US8609852, 4)
Affinity DataKi:  2.60nM ΔG°:  -49.0kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109097BDBM109097(US8609852, 3)
Affinity DataKi:  2.70nM ΔG°:  -48.9kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109112BDBM109112(US8609852, 19)
Affinity DataKi:  2.80nM ΔG°:  -48.8kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109169BDBM109169(US8609852, 76)
Affinity DataKi:  3nM ΔG°:  -48.6kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109184BDBM109184(US8609852, 93)
Affinity DataKi:  3nM ΔG°:  -48.6kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 50123009BDBM50123009(CHEMBL332396 | US8609852, 80 | 3-Methyl-5-(2-methy...)
Affinity DataKi:  3nM ΔG°:  -48.6kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109129BDBM109129(US8609852, 36)
Affinity DataKi:  3nM ΔG°:  -48.6kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109110BDBM109110(US8609852, 17)
Affinity DataKi:  3.80nM ΔG°:  -48.1kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109152BDBM109152(US8609852, 59)
Affinity DataKi:  4nM ΔG°:  -47.9kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109168BDBM109168(US8609852, 75)
Affinity DataKi:  4nM ΔG°:  -47.9kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109156BDBM109156(US8609852, 63)
Affinity DataKi:  4nM ΔG°:  -47.9kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109181BDBM109181(US8609852, 90)
Affinity DataKi:  4nM ΔG°:  -47.9kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109132BDBM109132(US8609852, 39)
Affinity DataKi:  4nM ΔG°:  -47.9kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109148BDBM109148(US8609852, 55)
Affinity DataKi:  4nM ΔG°:  -47.9kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109179BDBM109179(US8609852, 88)
Affinity DataKi:  4nM ΔG°:  -47.9kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109164BDBM109164(US8609852, 71)
Affinity DataKi:  4.5nM ΔG°:  -47.6kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

TargetMetabotropic glutamate receptor 5(Rat)
Merck Sharp & Dohme

US Patent
LigandChemical structure of BindingDB Monomer ID 109125BDBM109125(US8609852, 32)
Affinity DataKi:  4.80nM ΔG°:  -47.5kJ/moleT: 2°CAssay Description:Binding assays were performed as described in Schaffhauser H, Richards J G, Cartmell J, Chaboz S, Kemp J A, Klingelschmidt A, Messer J, Stadler H, Wo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2014
Entry Details
US Patent

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