Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 7127
TargetMitogen-activated protein kinase 1 [L114A](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176676(US9115122, 2.3.2)
Affinity DataKd:  27nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [L235A](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176676(US9115122, 2.3.2)
Affinity DataKd:  90nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [L232A](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176676(US9115122, 2.3.2)
Affinity DataKd:  130nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176676(US9115122, 2.3.2)
Affinity DataKd:  130nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [Y191A](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176676(US9115122, 2.3.2)
Affinity DataKd:  130nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [L198A,L232A](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176676(US9115122, 2.3.2)
Affinity DataKd:  140nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176678(US9115122, SF-2-054)
Affinity DataKd:  170nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [R275A](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176676(US9115122, 2.3.2)
Affinity DataKd:  240nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [L265A](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176676(US9115122, 2.3.2)
Affinity DataKd:  280nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176678(US9115122, SF-2-054)
Affinity DataKd:  400nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176677(US9115122, SF-2-062)
Affinity DataKd:  1.30E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176678(US9115122, SF-2-054)
Affinity DataKd:  1.40E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176674(US9115122, 76.3)
Affinity DataKd:  1.50E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [D319N](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176673(US9115122, 76.2)
Affinity DataKd:  1.90E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176675(US9115122, 76.4)
Affinity DataKd:  2.40E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [T157A](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176673(US9115122, 76.2)
Affinity DataKd:  2.40E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [T157A](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176675(US9115122, 76.4)
Affinity DataKd:  3.00E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176673(US9115122, 76.2)
Affinity DataKd:  3.30E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176677(US9115122, SF-2-062)
Affinity DataKd:  3.70E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [T157A,D319N](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176673(US9115122, 76.2)
Affinity DataKd:  4.00E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176677(US9115122, SF-2-062)
Affinity DataKd:  4.20E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176674(US9115122, 76.3)
Affinity DataKd:  4.50E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176672(US9115122, 76)
Affinity DataKd:  5.00E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176677(US9115122, SF-2-062)
Affinity DataKd:  6.00E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [T157A](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176672(US9115122, 76)
Affinity DataKd:  6.10E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [T157A,D319N](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176672(US9115122, 76)
Affinity DataKd:  6.40E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176677(US9115122, SF-2-062)
Affinity DataKd:  6.80E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [D319N](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176672(US9115122, 76)
Affinity DataKd:  7.00E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176672(US9115122, 76)
Affinity DataKd:  7.00E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [T157A](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176674(US9115122, 76.3)
Affinity DataKd:  8.10E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176679(US9115122, SS-1-019)
Affinity DataKd:  8.30E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176679(US9115122, SS-1-019)
Affinity DataKd:  9.30E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176678(US9115122, SF-2-054)
Affinity DataKd:  1.02E+4nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176678(US9115122, SF-2-054)
Affinity DataKd:  1.20E+4nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [D319N](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176674(US9115122, 76.3)
Affinity DataKd:  1.34E+4nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [D319N](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176675(US9115122, 76.4)
Affinity DataKd:  1.80E+4nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [L198A,L235A](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176676(US9115122, 2.3.2)
Affinity DataKd: >2.00E+4nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [T157A,D319N](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176674(US9115122, 76.3)
Affinity DataKd: >2.00E+4nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent

TargetMitogen-activated protein kinase 1 [T157A,D319N](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176675(US9115122, 76.4)
Affinity DataKd: >2.00E+4nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
US Patent