Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 8307
TargetPolyphenol oxidase 1(White button mushroom)
Pierre Fabre Dermo-Cosmetique

US Patent
LigandPNGBDBM240726(US9422261, Compound 4)
Affinity DataIC50: 80nMpH: 6.8Assay Description:Reader: Synergy HT program: tyrosinase 280-490 kinetics: kinetics over 45 minutes, reading at t=10 minutes, Tests in transparent 96-well plates, Phos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

TargetPolyphenol oxidase 1(White button mushroom)
Pierre Fabre Dermo-Cosmetique

US Patent
LigandPNGBDBM240723(US9422261, Compound 1)
Affinity DataIC50: 90nMpH: 6.8Assay Description:Reader: Synergy HT program: tyrosinase 280-490 kinetics: kinetics over 45 minutes, reading at t=10 minutes, Tests in transparent 96-well plates, Phos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

TargetPolyphenol oxidase 1(White button mushroom)
Pierre Fabre Dermo-Cosmetique

US Patent
LigandPNGBDBM240731(US9422261, 4-(1- phenylethyl) benzene-1,3- diol)
Affinity DataIC50: 100nMpH: 6.8Assay Description:Reader: Synergy HT program: tyrosinase 280-490 kinetics: kinetics over 45 minutes, reading at t=10 minutes, Tests in transparent 96-well plates, Phos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

TargetPolyphenol oxidase 1(White button mushroom)
Pierre Fabre Dermo-Cosmetique

US Patent
LigandPNGBDBM240725(US9422261, Compound 3)
Affinity DataIC50: 200nMpH: 6.8Assay Description:Reader: Synergy HT program: tyrosinase 280-490 kinetics: kinetics over 45 minutes, reading at t=10 minutes, Tests in transparent 96-well plates, Phos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

TargetPolyphenol oxidase 1(White button mushroom)
Pierre Fabre Dermo-Cosmetique

US Patent
LigandPNGBDBM240724(US9422261, Compound 2)
Affinity DataIC50: 400nMpH: 6.8Assay Description:Reader: Synergy HT program: tyrosinase 280-490 kinetics: kinetics over 45 minutes, reading at t=10 minutes, Tests in transparent 96-well plates, Phos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

TargetPolyphenol oxidase 1(White button mushroom)
Pierre Fabre Dermo-Cosmetique

US Patent
LigandPNGBDBM50248158(N-butylresorcinol | CHEMBL450195 | US8993596, 4-Bu...)
Affinity DataIC50: 1.00E+3nMpH: 6.8Assay Description:Reader: Synergy HT program: tyrosinase 280-490 kinetics: kinetics over 45 minutes, reading at t=10 minutes, Tests in transparent 96-well plates, Phos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

TargetPolyphenol oxidase 1(White button mushroom)
Pierre Fabre Dermo-Cosmetique

US Patent
LigandPNGBDBM240727(US9422261, Compound 5)
Affinity DataIC50: 1.50E+3nMpH: 6.8Assay Description:Reader: Synergy HT program: tyrosinase 280-490 kinetics: kinetics over 45 minutes, reading at t=10 minutes, Tests in transparent 96-well plates, Phos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

TargetPolyphenol oxidase 1(White button mushroom)
Pierre Fabre Dermo-Cosmetique

US Patent
LigandPNGBDBM240729(US9422261, Unigen resorcinol derivative | US968291...)
Affinity DataIC50: 2.00E+3nMpH: 6.8Assay Description:Reader: Synergy HT program: tyrosinase 280-490 kinetics: kinetics over 45 minutes, reading at t=10 minutes, Tests in transparent 96-well plates, Phos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

TargetPolyphenol oxidase 1(White button mushroom)
Pierre Fabre Dermo-Cosmetique

US Patent
LigandPNGBDBM240730(US9422261, Unigen resorcinol derivative | US968291...)
Affinity DataIC50: 4.90E+3nMpH: 6.8Assay Description:Reader: Synergy HT program: tyrosinase 280-490 kinetics: kinetics over 45 minutes, reading at t=10 minutes, Tests in transparent 96-well plates, Phos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

TargetPolyphenol oxidase 1(White button mushroom)
Pierre Fabre Dermo-Cosmetique

US Patent
LigandPNGBDBM50031467(Kojic Acid | CHEMBL287556 | 5-HYDROXY-2-(HYDROXYME...)
Affinity DataIC50: 1.50E+4nMpH: 6.8Assay Description:Reader: Synergy HT program: tyrosinase 280-490 kinetics: kinetics over 45 minutes, reading at t=10 minutes, Tests in transparent 96-well plates, Phos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

TargetPolyphenol oxidase 1(White button mushroom)
Pierre Fabre Dermo-Cosmetique

US Patent
LigandPNGBDBM240728(US9422261, Arbutin)
Affinity DataIC50: 9.00E+4nMpH: 6.8Assay Description:Reader: Synergy HT program: tyrosinase 280-490 kinetics: kinetics over 45 minutes, reading at t=10 minutes, Tests in transparent 96-well plates, Phos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent