Compile Data Set for Download or QSAR
Report error Found 173 Enz. Inhib. hit(s) with all data for entry = 1841
TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343230BDBM343230(1-methyl-4-(5-methylpyridin-2-yl)-N-(2-phenylimida...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343231BDBM343231(1-methyl-4-(4-methylthiazol-2-yl)-N-(2-phenylimida...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343234BDBM343234(1-methyl-N-(2-phenylimidazo[1,2-a]pyridin-7-yl)-4-...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343235BDBM343235(1-methyl-N-(2-phenylimidazo[1,2-a]pyridin-7-yl)-4-...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343232BDBM343232(4-(4-(difluoromethyl)thiazol-2-yl)-1-methyl-N-(2-p...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343233BDBM343233(4-(4-(difluoromethyl)-5-methylthiazol-2-yl)-1-meth...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343237BDBM343237(1-methyl-4-(5-methyl-1,3,4-thiadiazol-2-yl)-N-(2-p...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343247BDBM343247(4-(6-methoxypyridin-2-yl)-1-methyl-N-(2-phenyl-5,6...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343244BDBM343244(N-(2-(3-fluorophenyl)-5,6,7,8-tetrahydroimidazo[1,...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343245BDBM343245(1-methyl-4-(6-methylpyridin-2-yl)-N-(2-phenyl-5,6,...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343250BDBM343250(4-(3-isopropyl-1,2,4-thiadiazol-5-yl)-1-methyl-N-(...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343251BDBM343251(1-methyl-4-(5-methylthiazol-2-yl)-N-(2-phenyl-5,6,...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343248BDBM343248(1-methyl-4-(2-methylthiazol-4-yl)-N-(2-phenyl-5,6,...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343249BDBM343249(1-methyl-4-(6-methylpyrazin-2-yl)-N-(2-phenyl-5,6,...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343238BDBM343238(4-(4-(difluoromethyl)thiazol-2-yl)-N-(2-(3-fluorop...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343239BDBM343239(1-methyl-N-(2-phenyl-5,6,7,8-tetrahydroimidazo[1,2...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343236BDBM343236(4-(5-chloro-4-(difluoromethyl)thiazol-2-yl)-1-meth...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343237BDBM343237(1-methyl-4-(5-methyl-1,3,4-thiadiazol-2-yl)-N-(2-p...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343242BDBM343242(4-(4-(difluoromethyl)-5-methylthiazol-2-yl)-1-meth...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343243BDBM343243(4-(4-(difluoromethyl)-5-methylthiazol-2-yl)-N-(2-(...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343240BDBM343240(4-(4-(difluoromethyl)thiazol-2-yl)-1-methyl-N-(2-p...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343241BDBM343241(4-(5-chloro-4-(difluoromethyl)thiazol-2-yl)-1-meth...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343266BDBM343266(N-(6-fluoro-2-phenyl-[1,2,4]triazolo[1,5-a]pyridin...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343267BDBM343267(US9777000, Example 3.20 | 4-(5-chloro-4-(difluorom...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343264BDBM343264(4-(4-(difluoromethyl)thiazol-2-yl)-N-(2-(4-fluorop...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343265BDBM343265(N-(2-(4-fluorophenyl)-5,6,7,8-tetrahydroimidazo[1,...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343255BDBM343255(N-(3-fluoro-2-phenyl-5,6,7,8-tetrahydroimidazo[1,2...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343258BDBM343258(1-methyl-4-(4-methylpyridin-2-yl)-N-(2-phenyl-5,6,...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343238BDBM343238(4-(4-(difluoromethyl)thiazol-2-yl)-N-(2-(3-fluorop...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343278BDBM343278(4-(3-cyanopyridin-2-yl)-N-(6-fluoro-2-phenyl-[1,2,...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343279BDBM343279(4-(3,6-dimethyl-pyrazin-2-yl)-N-(6-fluoro-2-phenyl...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343276BDBM343276(4-(4,6-dimethylpyridin-2-yl)-N-(6-fluoro-2-phenyl-...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343277BDBM343277(4-(4-(difluoromethyl)thiazol-2-yl)-N-(6-fluoro-2-p...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343282BDBM343282(4-(4-(difluoromethyl)thiazol-2-yl)-N-(2-(3-fluorop...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343283BDBM343283(4-(4-ethylthiazol-2-yl)-1-methyl-N-(2-phenyl-[1,2,...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343280BDBM343280(4-(4-(difluoromethyl)thiazol-2-yl)-1-methyl-N-(2-p...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343281BDBM343281(4-(4-(difluoromethyl)thiazol-2-yl)-N-(2-(2-methoxy...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343270BDBM343270(US9777000, Example 3.50 | 4-(2,5-dimethylpyrimidin...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343271BDBM343271(N-(6-fluoro-2-phenyl-[1,2,4]triazolo[1,5-a]pyridin...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343268BDBM343268(US9777000, Example 3.30 | 4-(2,6-dimethylpyrimidin...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343269BDBM343269(US9777000, Example 3.40 | 4-(2,6-dimethoxypyrimidi...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343274BDBM343274(N-(6-fluoro-2-phenyl-[1,2,4]triazolo[1,5-a]pyridin...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343266BDBM343266(N-(6-fluoro-2-phenyl-[1,2,4]triazolo[1,5-a]pyridin...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343272BDBM343272(N-(6-fluoro-2-phenyl-[1,2,4]triazolo[1,5-a]pyridin...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343273BDBM343273(N-(6-fluoro-2-phenyl-[1,2,4]triazolo[1,5-a]pyridin...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343294BDBM343294(4-(5-chloropyrimidin-4-yl)-N-(6-fluoro-2-phenyl-[1...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343268BDBM343268(US9777000, Example 3.30 | 4-(2,6-dimethylpyrimidin...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343292BDBM343292(4-(5-fluoro-2-methoxypyrimidin-4-yl)-N-(6-fluoro-2...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343293BDBM343293(N-(6-fluoro-2-phenyl-[1,2,4]triazolo[1,5-a]pyridin...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Mochida Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 343298BDBM343298(N-(6-fluoro-2-phenyl-[1,2,4]triazolo[1,5-a]pyridin...)
Affinity DataIC50: 5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details
US Patent

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