Reaction Details Report a problem with these data
Target
Protein kinase C beta type Isoform 2
Ligand
BDBM533459
Substrate
n/a
Meas. Tech.
Protein Kinase C beta 2 (PKCpII) Assay
Ki
1.17±n/a nM
Citation
Li, H; Nukui, S; Scales, SA; Teng, M; Yin, C Substituted N-pyrimidin-4-yl-3-aminopyrrolo[3,4-C]pyrazoles as protein kinase C inhibitors US Patent US11780853 Publication Date 10/10/2023
More Info.:
Target
Name:
Isoform Beta-II of Protein kinase C beta type (PRKCB2)
Synonyms:
KPCB_HUMAN | PKCB | PRKCB | PRKCB1 | Protein kinase C beta II type | Protein kinase C beta type (PRKCB2)
Type:
Enzyme
Mol. Mass.:
77017.33
Organism:
Human
Description:
P05771-2
Residue:
673
Sequence:
MADPAAGPPPSEGEESTVRFARKGALRQKNVHEVKNHKFTARFFKQPTFCSHCTDFIWGFGKQGFQCQVCCFVVHKRCHEFVTFSCPGADKGPASDDPRSKHKFKIHTYSSPTFCDHCGSLLYGLIHQGMKCDTCMMNVHKRCVMNVPSLCGTDHTERRGRIYIQAHIDRDVLIVLVRDAKNLVPMDPNGLSDPYVKLKLIPDPKSESKQKTKTIKCSLNPEWNETFRFQLKESDKDRRLSVEIWDWDLTSRNDFMGSLSFGISELQKASVDGWFKLLSQEEGEYFNVPVPPEGSEANEELRQKFERAKISQGTKVPEEKTTNTVSKFDNNGNRDRMKLTDFNFLMVLGKGSFGKVMLSERKGTDELYAVKILKKDVVIQDDDVECTMVEKRVLALPGKPPFLTQLHSCFQTMDRLYFVMEYVNGGDLMYHIQQVGRFKEPHAVFYAAEIAIGLFFLQSKGIIYRDLKLDNVMLDSEGHIKIADFGMCKENIWDGVTTKTFCGTPDYIAPEIIAYQPYGKSVDWWAFGVLLYEMLAGQAPFEGEDEDELFQSIMEHNVAYPKSMSKEAVAICKGLMTKHPGKRLGCGPEGERDIKEHAFFRYIDWEKLERKEIQPPYKPKACGRNAENFDRFFTRHPPVLTPPDQEVIRNIDQSEFEGFSFVNSEFLKPEVKS