Reaction Details Report a problem with these data
Target
Melatonin receptor
Ligand
BDBM82556
Substrate
n/a
Ki
460±n/a nM
Comments
PDSP_7421
Citation
 Morgan, PJ; Barrett, P; Howell, HE; Helliwell, R Melatonin receptors: localization, molecular pharmacology and physiological significance. Neurochem Int 24:101-46 (1994) [PubMed]  Article 
Target
Name:
Melatonin receptor
Synonyms:
Melatonin | Melatonin receptor
Type:
Enzyme Catalytic Domain
Mol. Mass.:
13287.02
Organism:
Rabbit
Description:
Q9BE38
Residue:
114
Sequence:
MIWMLTLVAVMPNLHTGTLQYDPRVYSCTFSQSVSSAYTIAVVVFHFIIPMLMSSCCYLRIWILVLQVRRRVKPDNKPKLKPQDFRNFITMFVVFVLFAICWAPLNFIVLLGRS
  
Inhibitor
Name:
BDBM82556
Synonyms:
melatonin, 6-Methoxy
Type:
Small organic molecule
Emp. Form.:
C14H18N2O3
Mol. Mass.:
262.3043
SMILES:
COc1cc2[nH]cc(CCNC(C)=O)c2cc1OC
Structure:
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