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Found 76 with Last Name = 'barrett' and Initial = 'p'
TargetMelatonin receptor(RABBIT)
Rowett Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM29611(2-Iodomelatonin | CHEMBL289233 | Melatonin,2-Iodo)
Affinity DataKi:  2.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor(RABBIT)
Rowett Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50043289(CHEMBL34730 | N-[2-(6-Chloro-5-methoxy-1H-indol-3-...)
In DepthDetails ArticlePubMed
TargetMelatonin receptor(RABBIT)
Rowett Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  6.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50148767(2,3-dihydroxy-4-(hydroxyamino)-4-oxobutyl dihydrog...)
Affinity DataKi:  10nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of Trypanosoma brucei expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50148780(((4R,5R)-5-(hydroxycarbamoyl)-2,2-dimethyl-1,3-dio...)
Affinity DataKi:  35nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of Trypanosoma brucei expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetMelatonin receptor(RABBIT)
Rowett Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM82509(Melatonin,6-Hydroxy | melatonin, 6-Hydroxy)
Affinity DataKi:  74nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50148765(1-(hydroxyamino)-1-oxo-4-(phosphonooxy)butane-2,3-...)
Affinity DataKi:  80nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of Trypanosoma brucei expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50148790((2R,3R)-2,3-Dihydroxy-4-phosphonooxy-butyric acid ...)
Affinity DataKi:  130nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of Trypanosoma brucei expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105135(CHEMBL542936 | N2-(3-((12-((3-((4Amino,6-(methylam...)
Affinity DataKi:  135nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105123(CHEMBL544581 | N2-(3-((12-((3-((4Amino,6-(dimethyl...)
Affinity DataKi:  240nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50148765(1-(hydroxyamino)-1-oxo-4-(phosphonooxy)butane-2,3-...)
Affinity DataKi:  360nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of sheep liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target6-phosphogluconate dehydrogenase, decarboxylating(Ovis aries)
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50148765(1-(hydroxyamino)-1-oxo-4-(phosphonooxy)butane-2,3-...)
Affinity DataKi:  360nMAssay Description:Inhibition of sheep 6PGDH expressed in Escherichia coli by spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105120(CHEMBL542932 | N-{3-[12-(3-Amino-propylamino)-dode...)
Affinity DataKi:  410nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor(RABBIT)
Rowett Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM82556(melatonin, 6-Methoxy)
Affinity DataKi:  460nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105124(CHEMBL553117 | N2-(3-[12-(3-[(4,6-Diamino-1,3,5-tr...)
Affinity DataKi:  500nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105137(CHEMBL545281 | N-{3-[12-(3-Amino-propylamino)-dode...)
Affinity DataKi:  600nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105121(CHEMBL542204 | N2-(3-((9-((3-((4-Amino-6-(methylam...)
Affinity DataKi:  750nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105125(CHEMBL541322 | N-{3-[12-(3-Amino-propylamino)-dode...)
Affinity DataKi:  1.00E+3nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target6-phosphogluconate dehydrogenase, decarboxylating(Ovis aries)
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50148780(((4R,5R)-5-(hydroxycarbamoyl)-2,2-dimethyl-1,3-dio...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of sheep 6PGDHMore data for this Ligand-Target Pair
Target6-phosphogluconate dehydrogenase, decarboxylating(Ovis aries)
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50148780(((4R,5R)-5-(hydroxycarbamoyl)-2,2-dimethyl-1,3-dio...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of sheep 6PGDH expressed in Escherichia coli by spectroscopyMore data for this Ligand-Target Pair
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50148780(((4R,5R)-5-(hydroxycarbamoyl)-2,2-dimethyl-1,3-dio...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of sheep liverMore data for this Ligand-Target Pair
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50148769((R)-Phosphoric acid mono-((R)-3-carbamoyl-2,3-dihy...)
Affinity DataKi:  1.52E+3nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of Trypanosoma brucei expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor(RABBIT)
Rowett Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50282758(CHEMBL33171 | N-Acetyltryptamine | N-[2-(1H-Indol-...)
Affinity DataKi:  1.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105139(CHEMBL544580 | N1,N9-Di(3-(((4,6-(dimethylamino-1,...)
Affinity DataKi:  2.40E+3nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105132(CHEMBL544335 | N2-(3-((12-((3-((4,6-Di(dimethylami...)
Affinity DataKi:  2.50E+3nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50148767(2,3-dihydroxy-4-(hydroxyamino)-4-oxobutyl dihydrog...)
Affinity DataKi:  2.54E+3nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of sheep liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target6-phosphogluconate dehydrogenase, decarboxylating(Ovis aries)
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50148767(2,3-dihydroxy-4-(hydroxyamino)-4-oxobutyl dihydrog...)
Affinity DataKi:  2.54E+3nMAssay Description:Inhibition of sheep 6PGDH expressed in Escherichia coli by spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor(RABBIT)
Rowett Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM29612(CHEMBL33103 | CVD-0001578 | JOH-MSK-a63bdd1d-4 | N...)
Affinity DataKi:  3.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105141(CHEMBL542698 | N2-(3-((12-((3-((4,6-Di(methylamino...)
Affinity DataKi:  3.20E+3nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50148777(2,3,4,5-tetrahydroxy-6-{[hydroxy(dioxido)phosphora...)
Affinity DataKi:  3.50E+3nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of Trypanosoma brucei expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50148786(3,4,5-trihydroxy-6-{[hydroxy(dioxido)phosphoranyl]...)
Affinity DataKi:  4.40E+3nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of Trypanosoma brucei expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor(RABBIT)
Rowett Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM82087(2-(5-methoxy-1H-indol-3-yl)ethanamine | 5-MT | 5-M...)
Affinity DataKi:  4.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105133(CHEMBL541581 | N1,N9-Di(3-(((4-amino-6-(dimethylam...)
Affinity DataKi:  4.60E+3nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105134(CHEMBL555240 | N1,N9-Di(3-(di((4,6-diamino-1,3,5-t...)
Affinity DataKi:  6.70E+3nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105119(CHEMBL539797 | N2-(3-((9-((3-((4-Amino-6-(methylam...)
Affinity DataKi:  1.00E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor(RABBIT)
Rowett Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50047013(2-(5-Methoxy-1H-indol-3-yl)-ethanol (5-methoxytryp...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50148790((2R,3R)-2,3-Dihydroxy-4-phosphonooxy-butyric acid ...)
Affinity DataKi:  1.07E+4nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of sheep liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target6-phosphogluconate dehydrogenase, decarboxylating(Ovis aries)
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50148790((2R,3R)-2,3-Dihydroxy-4-phosphonooxy-butyric acid ...)
Affinity DataKi:  1.08E+4nMAssay Description:Inhibition of sheep 6PGDH expressed in Escherichia coli by spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105129(CHEMBL542208 | N2-(3-((9-((3-((4,6-Di(methylamino)...)
Affinity DataKi:  1.40E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50148777(2,3,4,5-tetrahydroxy-6-{[hydroxy(dioxido)phosphora...)
Affinity DataKi:  1.60E+4nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of sheep liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105142(CHEMBL554895 | N-{3-[9-(3-Amino-propylamino)-nonyl...)
Affinity DataKi:  1.70E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105118(CHEMBL536324 | N1,N9-Di(3-(((4-amino-6-(dimethylam...)
Affinity DataKi:  1.70E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105138(CHEMBL543641 | N2-(3-[9-(3-[(4,6-Diamino-1,3,5-tri...)
Affinity DataKi:  1.90E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105128(CHEMBL538778 | N-{3-[12-(3-Amino-propylamino)-dode...)
Affinity DataKi:  2.50E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105143(CHEMBL544116 | N2-(3-((9-((3-((4,6-Di(dimethylamin...)
Affinity DataKi:  2.90E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105131(CHEMBL553511 | N1,N9-Di(3-(((4,6-(dimethylamino-1,...)
Affinity DataKi:  3.00E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50148769((R)-Phosphoric acid mono-((R)-3-carbamoyl-2,3-dihy...)
Affinity DataKi:  3.92E+4nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of sheep liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50148785(((R)-2-Acetoxy-3-phosphonooxy-propane-1-sulfinyl)-...)
Affinity DataKi:  4.00E+4nMAssay Description:Inhibition constant against 6-phosphogluconate dehydrogenase of Trypanosoma brucei expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105136(CHEMBL552613 | N2-(3-[2-(3-[(4,6-Diamino-1,3,5-tri...)
Affinity DataKi:  5.50E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target6-phosphogluconate dehydrogenase, decarboxylating(Ovis aries)
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50322321(5-phospho-D-ribonate | CHEMBL1173785)
Affinity DataKi:  6.65E+4nMAssay Description:Inhibition of sheep 6PGDH expressed in Escherichia coli by spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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