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Target
Probable G-protein coupled receptor 34
Ligand
BDBM50238945
Substrate
n/a
Meas. Tech.
ChEMBL_1664555 (CHEMBL4014236)
EC50
>3000±n/a nM
Citation
Sayama, M; Sayama, M; Sayama, M; Inoue, A; Inoue, A; Inoue, A; Nakamura, S; Nakamura, S; Nakamura, S; Jung, S; Jung, S; Jung, S; Ikubo, M; Ikubo, M; Ikubo, M; Otani, Y; Otani, Y; Otani, Y; Uwamizu, A; Uwamizu, A; Uwamizu, A; Kishi, T; Kishi, T; Kishi, T; Makide, K; Makide, K; Makide, K; Aoki, J; Aoki, J; Aoki, J; Hirokawa, T; Hirokawa, T; Hirokawa, T; Ohwada, T; Ohwada, T; Ohwada, T Probing the Hydrophobic Binding Pocket of G-Protein-Coupled Lysophosphatidylserine Receptor GPR34/LPS J Med Chem 60:6384-6399 (2017) [PubMed] Article
More Info.:
Target
Name:
Probable G-protein coupled receptor 34
Synonyms:
G protein-coupled receptor 34 | GPR34_MOUSE | Gpr34 | Probable G-protein coupled receptor 34
Type:
PROTEIN
Mol. Mass.:
43201.40
Organism:
Mus musculus
Description:
ChEMBL_102842
Residue:
375
Sequence:
MTTTSVDSWLCSSHGMHFITNYSDQASQNFSGVPNVTSCPMDEKLLSTVLTTFYSVIFLVGLVGNIIALYVFLGIHRKRNSIQIYLLNVAVADLLLIFCLPFRIMYHINQNKWTLGVILCKVVGTLFYMNMYISIILLGFISLDRYIKINRSIQQRRAITTKQSIYVCCIVWTVALAGFLTMIILTLKKGGHNSTMCFHYRDRHNAKGEAIFNFVLVVMFWLIFLLIILSYIKIGKNLLRISKRRSKFPNSGKYATTARNSFIVLIIFTICFVPYHAFRFIYISSQLNVSSCYWKEIIHKTNEIMLVFSSFNSCLDPVMYFLMSSNIRKIMCQLLFRRFQSEASRSESTSEFKPGHSLHDLSVTVKMPQYSTKGN