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Target
Probable G-protein coupled receptor 34
Ligand
BDBM50096422
Substrate
n/a
Meas. Tech.
ChEMBL_1664555 (CHEMBL4014236)
EC50
>3162±n/a nM
Citation
 Sayama, M; Sayama, M; Sayama, M; Inoue, A; Inoue, A; Inoue, A; Nakamura, S; Nakamura, S; Nakamura, S; Jung, S; Jung, S; Jung, S; Ikubo, M; Ikubo, M; Ikubo, M; Otani, Y; Otani, Y; Otani, Y; Uwamizu, A; Uwamizu, A; Uwamizu, A; Kishi, T; Kishi, T; Kishi, T; Makide, K; Makide, K; Makide, K; Aoki, J; Aoki, J; Aoki, J; Hirokawa, T; Hirokawa, T; Hirokawa, T; Ohwada, T; Ohwada, T; Ohwada, T Probing the Hydrophobic Binding Pocket of G-Protein-Coupled Lysophosphatidylserine Receptor GPR34/LPS J Med Chem 60:6384-6399 (2017) [PubMed]  Article 
Target
Name:
Probable G-protein coupled receptor 34
Synonyms:
G protein-coupled receptor 34 | GPR34_MOUSE | Gpr34 | Probable G-protein coupled receptor 34
Type:
PROTEIN
Mol. Mass.:
43201.40
Organism:
Mus musculus
Description:
ChEMBL_102842
Residue:
375
Sequence:
MTTTSVDSWLCSSHGMHFITNYSDQASQNFSGVPNVTSCPMDEKLLSTVLTTFYSVIFLVGLVGNIIALYVFLGIHRKRNSIQIYLLNVAVADLLLIFCLPFRIMYHINQNKWTLGVILCKVVGTLFYMNMYISIILLGFISLDRYIKINRSIQQRRAITTKQSIYVCCIVWTVALAGFLTMIILTLKKGGHNSTMCFHYRDRHNAKGEAIFNFVLVVMFWLIFLLIILSYIKIGKNLLRISKRRSKFPNSGKYATTARNSFIVLIIFTICFVPYHAFRFIYISSQLNVSSCYWKEIIHKTNEIMLVFSSFNSCLDPVMYFLMSSNIRKIMCQLLFRRFQSEASRSESTSEFKPGHSLHDLSVTVKMPQYSTKGN
  
Inhibitor
Name:
BDBM50096422
Synonyms:
CHEMBL3577137
Type:
Small organic molecule
Emp. Form.:
C24H46NO8P
Mol. Mass.:
507.5977
SMILES:
CCCCCCCC\C=C/CCCCCCCC(=O)OCCCOP(O)(=O)OC[C@H](N)C(O)=O |r|
Structure:
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