Reaction Details
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Target
Genome polyprotein
Ligand
BDBM123409
Substrate
n/a
Meas. Tech.
Inhibition Assay
pH
7.5±n/a
Temperature
303.15±n/a K
Ki
1000±n/a nM
Comments
extracted
Citation
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More Info.:
Target
Name:
Genome polyprotein
Synonyms:
NS3-4A protease
Type:
Enzyme
Mol. Mass.:
72788.46
Organism:
Hepatitis C virus
Description:
K7XGM7
Residue:
681
Sequence:
APTAYAQQTRGLLGCITSLTGRDKNQVEGEVQIVSTAAQTFLATCINGVCWTVYHGAGTRTIASPKGPVIQMYTNVDKDLVGWPAPQGARSLTPCCGSSDLYLVTRHADVIPVRRRGDRGSLLSPRPISYLKGSSGGPLLCPAGHAVGIFRAAVCTRGVAKAVDFIPVESLETTMRSPVFTDNSSPPAVPQSFQVAHLHAPTGSGKSTRVPAAYAAQGYKVLVLNPSVAATLGFGAYMSKAHGVDPNVRTGVRTITTGSPITYSTYGKFLADGGCSGGAYDIIICDECHSTDATSILGIGTVLDQAETAGARLVVLATATPPGSVTVHPNIEEVALSTTGEIPFYGKAIPLEIKGGRHLIFCHSKKKCDELAAKLLGINAVAYYRGLDVSVIPTSGDVVVVATDALMTGFTGDFDSVIDCNTCVTQTVDFSLDPTFTLETTTLPQDAVRTQRRGRTGRGRPGIYRFVTPGERPSGMFDSSVLCECYDAGCAWYELTPAETTVRLRAYMNTPGLPVCQDHLEFWEGVFTGLTHIDAHFLSQTKQSGENLPYLVAYQATVCARAQAPPSWDQMWKCLRLKPTLHGPTPLLYRLGAVQNEITLTHPTKYIMTCMSADLEVVTSTWVLVGGVLAALAYCLSTGCVVIVGRIVLSGRPAIIPDREVLYEFDEMEECSQHLPYIEQG