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Target
Stimulator of interferon genes protein
Ligand
BDBM50509411
Substrate
n/a
Meas. Tech.
ChEMBL_1838268 (CHEMBL4338401)
EC50
20±n/a nM
Citation
Novotná, B; Vaneková, L; Zav?el, M; Bud??ínský, M; Dejmek, M; Smola, M; Gutten, O; Tehrani, ZA; Pimková Polidarová, M; Brázdová, A; Liboska, R; ?t?pánek, I; Vav?ina, Z; Jandu?ík, T; Nencka, R; Rulí?ek, L; Bou?a, E; Brynda, J; Páv, O; Birku?, G Enzymatic Preparation of 2'-5',3'-5'-Cyclic Dinucleotides, Their Binding Properties to Stimulator of Interferon Genes Adaptor Protein, and Structure/Activity Correlations. J Med Chem 62:10676-10690 (2019) [PubMed] Article
More Info.:
Target
Name:
Stimulator of interferon genes protein
Synonyms:
ERIS | Endoplasmic reticulum interferon stimulator | MITA | Mediator of IRF3 activation | STING | STING1 | STING_HUMAN | Synonyms=ERIS | TMEM173 | Transmembrane protein 173 | hMITA | hSTING
Type:
Protein
Mol. Mass.:
42195.64
Organism:
Human
Description:
Q86WV6
Residue:
379
Sequence:
MPHSSLHPSIPCPRGHGAQKAALVLLSACLVTLWGLGEPPEHTLRYLVLHLASLQLGLLLNGVCSLAEELRHIHSRYRGSYWRTVRACLGCPLRRGALLLLSIYFYYSLPNAVGPPFTWMLALLGLSQALNILLGLKGLAPAEISAVCEKGNFNVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQQTGDHAGIKDRVYSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCRTLEDILADAPESQNNCRLIAYQEPADDSSFSLSQEVLRHLRQEEKEEVTVGSLKTSAVPSTSTMSQEPELLISGMEKPLPLRTDFS