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Target
Polynucleotide kinase
Ligand
BDBM50356642
Substrate
n/a
Meas. Tech.
ChEMBL_785421 (CHEMBL1919800)
IC50
>100000±n/a nM
Citation
Maruo, S; Kuriyama, I; Kuramochi, K; Tsubaki, K; Yoshida, H; Mizushina, Y Inhibitory effect of novel 5-O-acyl juglones on mammalian DNA polymerase activity, cancer cell growth and inflammatory response. Bioorg Med Chem 19:5803-12 (2011) [PubMed] Article
More Info.:
Target
Name:
Polynucleotide kinase
Synonyms:
KIPN_BPT4 | pseT
Type:
PROTEIN
Mol. Mass.:
34626.48
Organism:
Enterobacteria phage T4
Description:
ChEMBL_1297302
Residue:
301
Sequence:
MKKIILTIGCPGSGKSTWAREFIAKNPGFYNINRDDYRQSIMAHEERDEYKYTKKKEGIVTGMQFDTAKSILYGGDSVKGVIISDTNLNPERRLAWETFAKEYGWKVEHKVFDVPWTELVKRNSKRGTKAVPIDVLRSMYKSMREYLGLPVYNGTPGKPKAVIFDVDGTLAKMNGRGPYDLEKCDTDVINPMVVELSKMYALMGYQIVVVSGRESGTKEDPTKYYRMTRKWVEDIAGVPLVMQCQREQGDTRKDDVVKEEIFWKHIAPHFDVKLAIDDRTQVVEMWRRIGVECWQVASGDF