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Target
Putative P2Y purinoceptor 10
Ligand
BDBM50096422
Substrate
n/a
Meas. Tech.
ChEMBL_1495909 (CHEMBL3579720)
EC50
25±n/a nM
Citation
Ikubo, M; Inoue, A; Nakamura, S; Jung, S; Sayama, M; Otani, Y; Uwamizu, A; Suzuki, K; Kishi, T; Shuto, A; Ishiguro, J; Okudaira, M; Kano, K; Makide, K; Aoki, J; Ohwada, T Structure-activity relationships of lysophosphatidylserine analogs as agonists of G-protein-coupled receptors GPR34, P2Y10, and GPR174. J Med Chem 58:4204-19 (2015) [PubMed] Article
More Info.:
Target
Name:
Putative P2Y purinoceptor 10
Synonyms:
P2RY10 | P2Y-like receptor | P2Y10 | P2Y10_HUMAN | Putative P2Y purinoceptor 10
Type:
PROTEIN
Mol. Mass.:
38793.96
Organism:
Human
Description:
ChEMBL_109762
Residue:
339
Sequence:
MANLDKYTETFKMGSNSTSTAEIYCNVTNVKFQYSLYATTYILIFIPGLLANSAALWVLCRFISKKNKAIIFMINLSVADLAHVLSLPLRIYYYISHHWPFQRALCLLCFYLKYLNMYASICFLTCISLQRCFFLLKPFRARDWKRRYDVGISAAIWIVVGTACLPFPILRSTDLNNNKSCFADLGYKQMNAVALVGMITVAELAGFVIPVIIIAWCTWKTTISLRQPPMAFQGISERQKALRMVFMCAAVFFICFTPYHINFIFYTMVKETIISSCPVVRIALYFHPFCLCLASLCCLLDPILYYFMASEFRDQLSRHGSSVTRSRLMSKESGSSMIG