Reaction Details Report a problem with these data
Target
Hrh3 protein
Ligand
BDBM22914
Substrate
n/a
Ki
3.981071705535±n/a nM
Comments
PDSP_1847
Citation
Barbier, AJ; Berridge, C; Dugovic, C; Laposky, AD; Wilson, SJ; Boggs, J; Aluisio, L; Lord, B; Mazur, C; Pudiak, CM; Langlois, X; Xiao, W; Apodaca, R; Carruthers, NI; Lovenberg, TW Acute wake-promoting actions of JNJ-5207852, a novel, diamine-based H3 antagonist. Br J Pharmacol 143:649-61 (2004) [PubMed] Article
More Info.:
Target
Name:
Hrh3 protein
Synonyms:
HISTAMINE H3 | HRH3 | Hrh3 protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
37860.96
Organism:
Rat
Description:
Q5PPG3
Residue:
344
Sequence:
MERAPPDGLMNASGTLAGEAAAAGGARGFSAAWTAVLAALMALLIVATVLGNALVMLAFVADSSLRTQNNFFLLNLAISDFLVGAFCIPLYVPYVLTGRWTFGRGLCKLWLVVDYLLCASSVFNIVLISYDRFLSVTRAVSYRAQQGDTRRAVRKMALVWVLAFLLYGPAILSWEYLSGGSSIPEGHCYAEFFYNWYFLITASTLEFFTPFLSVTFFNLSIYLNIQRRTRLRLDGGREAGPEPPPDAQPSPPPAPPSCWGCWPKGHGEAMPLHRGSKPSASSASLEKRMKMVSQSITQRFRLSRDKKVAKSLAIIVSIFGLCWAPYTLLMIIRAACHGRCIPDY