Reaction Details Report a problem with these data
Target
Solute carrier family 13 member 5
Ligand
BDBM610832
Substrate
n/a
Meas. Tech.
Assay of the Citric Acid Cycle Activation
EC50
62.0±n/a nM
Citation
Sato, S; Matsuda, S; Matsumura, C; Itotani, M; Shinohara, T; Fujita, S; Sakurai, Y; Tai, K; Fukushima, T; Kanemoto, N; Okamoto, T Cyanotriazole compounds US Patent US10626095 Publication Date 4/21/2020
More Info.:
Target
Name:
Solute carrier family 13 member 5
Synonyms:
NACT | Na(+)/citrate cotransporter | S13A5_HUMAN | SLC13A5 | Sodium-coupled citrate transporter | Sodium-dependent citrate transporter | Solute carrier family 13 member 5
Type:
PROTEIN
Mol. Mass.:
63069.06
Organism:
Homo sapiens (Human)
Description:
ChEMBL_116736
Residue:
568
Sequence:
MASALSYVSKFKSFVILFVTPLLLLPLVILMPAKFVRCAYVIILMAIYWCTEVIPLAVTSLMPVLLFPLFQILDSRQVCVQYMKDTNMLFLGGLIVAVAVERWNLHKRIALRTLLWVGAKPARLMLGFMGVTALLSMWISNTATTAMMVPIVEAILQQMEATSAATEAGLELVDKGKAKELPGSQVIFEGPTLGQQEDQERKRLCKAMTLCICYAASIGGTATLTGTGPNVVLLGQMNELFPDSKDLVNFASWFAFAFPNMLVMLLFAWLWLQFVYMRFNFKKSWGCGLESKKNEKAALKVLQEEYRKLGPLSFAEINVLICFFLLVILWFSRDPGFMPGWLTVAWVEGETKYVSDATVAIFVATLLFIVPSQKPKFNFRSQTEEERKTPFYPPPLLDWKVTQEKVPWGIVLLLGGGFALAKGSEASGLSVWMGKQMEPLHAVPPAAITLILSLLVAVFTECTSNVATTTLFLPIFASMSRSIGLNPLYIMLPCTLSASFAFMLPVATPPNAIVFTYGHLKVADMVKTGVIMNIIGVFCVFLAVNTWGRAIFDLDHFPDWANVTHIET