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Target
Zinc finger protein mex-5
Ligand
BDBM52790
Substrate
n/a
Meas. Tech.
Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2
EC50
96973±n/a nM
Citation
 PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2 PubChem Bioassay (2009)[AID] 
Target
Name:
Zinc finger protein mex-5
Synonyms:
MEX5_CAEEL | RecName: Full=Zinc finger protein mex-5 | mex-5
Type:
Enzyme Catalytic Domain
Mol. Mass.:
52832.78
Organism:
Caenorhabditis elegans
Description:
gi_55976631
Residue:
468
Sequence:
MKAASNSVSSAGGSVSPTTTQPPLPPGQSSHPQIYDQQMQYYFAAAMPNQPMATYAAQNGSSQQYAPAAPYYQDANGQYVQVPANGSMAPQQHMMVSGQPYLYMAQPQQGAQQVMQSGQPQLIYYQQSMAPQAAPMYFHPMQAAPMLPEQMGVMPHTQPAIPPQQQPRQVGVEISSTRTAPLTSSTPLPTSLEYETVQRDNRNRNIQFRYHRVMEHDELPIDEISKITLDNHNDDTMSAEKENHFHEHRGEKFGRRGFPIPETDSQQPPNYKTRLCMMHASGIKPCDMGARCKFAHGLKELRATDAPARYPNNKYKTKLCKNFARGGTGFCPYGLRCEFVHPTDKEFQNIPPYQRMSHDDQDYDQDVIPEDYVVARHQPRFMRTGGRATTPTKVMLKHRNVAGSMMCLSNAGRDLQAGGDYNQPESNEDDLPPHLRRNRRENPPMNKRRTSLSTKWTSEENLGLRGHY
  
Inhibitor
Name:
BDBM52790
Synonyms:
(3Z)-4-keto-2-[4-(3-phenylpropyl)pyridin-1-ium-1-yl]-3-(2-thienylsulfonylimino)naphthalen-1-olate | (3Z)-4-oxidanylidene-2-[4-(3-phenylpropyl)pyridin-1-ium-1-yl]-3-thiophen-2-ylsulfonylimino-naphthalen-1-olate | (3Z)-4-oxo-2-[4-(3-phenylpropyl)-1-pyridin-1-iumyl]-3-thiophen-2-ylsulfonylimino-1-naphthalenolate | (3Z)-4-oxo-2-[4-(3-phenylpropyl)pyridin-1-ium-1-yl]-3-thiophen-2-ylsulfonyliminonaphthalen-1-olate | MLS000768804 | SMR000433629 | cid_16412199
Type:
Small organic molecule
Emp. Form.:
C28H22N2O4S2
Mol. Mass.:
514.615
SMILES:
O=C1C([N-]S(=O)(=O)c2cccs2)=C(C(=O)c2ccccc12)[n+]1ccc(CCCc2ccccc2)cc1 |c:12|
Structure:
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