Reaction Details Report a problem with these data
Target
Zinc finger protein mex-5
Ligand
BDBM52807
Substrate
n/a
Meas. Tech.
Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2
EC50
300000±n/a nM
Citation
 PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2 PubChem Bioassay (2009)[AID] 
Target
Name:
Zinc finger protein mex-5
Synonyms:
MEX5_CAEEL | RecName: Full=Zinc finger protein mex-5 | mex-5
Type:
Enzyme Catalytic Domain
Mol. Mass.:
52832.78
Organism:
Caenorhabditis elegans
Description:
gi_55976631
Residue:
468
Sequence:
MKAASNSVSSAGGSVSPTTTQPPLPPGQSSHPQIYDQQMQYYFAAAMPNQPMATYAAQNGSSQQYAPAAPYYQDANGQYVQVPANGSMAPQQHMMVSGQPYLYMAQPQQGAQQVMQSGQPQLIYYQQSMAPQAAPMYFHPMQAAPMLPEQMGVMPHTQPAIPPQQQPRQVGVEISSTRTAPLTSSTPLPTSLEYETVQRDNRNRNIQFRYHRVMEHDELPIDEISKITLDNHNDDTMSAEKENHFHEHRGEKFGRRGFPIPETDSQQPPNYKTRLCMMHASGIKPCDMGARCKFAHGLKELRATDAPARYPNNKYKTKLCKNFARGGTGFCPYGLRCEFVHPTDKEFQNIPPYQRMSHDDQDYDQDVIPEDYVVARHQPRFMRTGGRATTPTKVMLKHRNVAGSMMCLSNAGRDLQAGGDYNQPESNEDDLPPHLRRNRRENPPMNKRRTSLSTKWTSEENLGLRGHY
  
Inhibitor
Name:
BDBM52807
Synonyms:
MLS000332823 | N-[3-Cyano-1-(3-ethoxy-propyl)-10-oxo-1,10-dihydro-1,9,10a-triaza-anthracen-(2Z)-ylidene]-acetamide | N-[3-cyano-1-(3-ethoxypropyl)-5-keto-dipyrido[1,2-d:3',4'-f]pyrimidin-2-ylidene]acetamide | N-[3-cyano-1-(3-ethoxypropyl)-5-oxidanylidene-dipyrido[1,2-d:3',4'-f]pyrimidin-2-ylidene]ethanamide | N-[3-cyano-1-(3-ethoxypropyl)-5-oxo-2-dipyrido[1,2-d:3',4'-f]pyrimidinylidene]acetamide | N-[3-cyano-1-(3-ethoxypropyl)-5-oxodipyrido[1,2-d:3',4'-f]pyrimidin-2-ylidene]acetamide | SMR000436199 | cid_1957999
Type:
Small organic molecule
Emp. Form.:
C19H19N5O3
Mol. Mass.:
365.3859
SMILES:
CCOCCCn1c2nc3ccccn3c(=O)c2cc(C#N)c1=NC(C)=O |w:23.26|
Structure:
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