Reaction Details Report a problem with these data
Target
Voltage-dependent calcium channel gamma-1 subunit
Ligand
BDBM81819
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_2652
Citation
Garritsen, A; Ijzerman, AP; Tulp, MT; Cragoe, EJ; Soudijn, W Receptor binding profiles of amiloride analogues provide no evidence for a link between receptors and the Na+/H+ exchanger, but indicate a common structure on receptor proteins. J Recept Res 11:891-907 (1991) [PubMed] Article
More Info.:
Target
Name:
Voltage-dependent calcium channel gamma-1 subunit
Synonyms:
CACNG1 | CACNLG | CCG1_HUMAN | Calcium channel (DHP) | Voltage-dependent calcium channel gamma-1 subunit
Type:
Enzyme Catalytic Domain
Mol. Mass.:
25030.69
Organism:
Homo sapiens (Human)
Description:
Calcium channel (DHP) 0 0::Q06432
Residue:
222
Sequence:
MSQTKMLKVRVTLFCILAGIVLAMTAVVTDHWAVLSPHMEHHNTTCEAAHFGLWRICTKRIPMDDSKTCGPITLPGEKNCSYFRHFNPGESSEIFEFTTQKEYSISAAAIAIFSLGFIILGSLCVLLSLGKKRDYLLRPASMFYAFAGLCILVSVEVMRQSVKRMIDSEDTVWIEYYYSWSFACACAAFILLFLGGLALLLFSLPRMPRNPWESCMDAEPEH