Reaction Details Report a problem with these data
Target
Cholecystokinin
Ligand
BDBM82232
Substrate
n/a
Ki
1000±n/a nM
Comments
PDSP_2616
Citation
 Van Dijk, A; Richards, JG; Trzeciak, A; Gillessen, D; Möhler, H Cholecystokinin receptors: biochemical demonstration and autoradiographical localization in rat brain and pancreas using [3H] cholecystokinin8 as radioligand. J Neurosci 4:1021-33 (1984) [PubMed] 
Target
Name:
Cholecystokinin
Synonyms:
CCKN_RAT | Cck
Type:
Enzyme Catalytic Domain
Mol. Mass.:
12844.29
Organism:
RAT
Description:
Cholecystokinin 0 RAT::P01355
Residue:
115
Sequence:
MKCGVCLCVVMAVLAAGALAQPVVPVEAVDPMEQRAEEAPRRQLRAVLRPDSEPRARLGALLARYIQQVRKAPSGRMSVLKNLQGLDPSHRISDRDYMGWMDFGRRSAEDYEYPS
  
Inhibitor
Name:
BDBM82232
Synonyms:
CAS_8977 | GDP | NSC_8977
Type:
Small organic molecule
Emp. Form.:
C10H15N5O11P2
Mol. Mass.:
443.2005
SMILES:
Nc1nc2n(cnc2c(=O)[nH]1)C1OC(COP(O)(=O)OP(O)(O)=O)C(O)C1O
Structure:
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