Reaction Details Report a problem with these data
Target
Adenosine receptor A3
Ligand
BDBM50258883
Substrate
n/a
Meas. Tech.
ChEBML_1690747
Ki
21±n/a nM
Citation
Azuaje, J; Jespers, W; Yaziji, V; Mallo, A; Majellaro, M; Caamaño, O; Loza, MI; Cadavid, MI; Brea, J; Åqvist, J; Sotelo, E; Gutiérrez-de-Terán, H Effect of Nitrogen Atom Substitution in A J Med Chem 60:7502-7511 (2017) [PubMed] Article
More Info.:
Target
Name:
Adenosine receptor A3
Synonyms:
A3 adenosine receptor (hA3) | AA3R_HUMAN | ADORA3 | Adenosine A3 receptor (A3AR)
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
36197.32
Organism:
Homo sapiens (Human)
Description:
P0DMS8
Residue:
318
Sequence:
MPNNSTALSLANVTYITMEIFIGLCAIVGNVLVICVVKLNPSLQTTTFYFIVSLALADIAVGVLVMPLAIVVSLGITIHFYSCLFMTCLLLIFTHASIMSLLAIAVDRYLRVKLTVRYKRVTTHRRIWLALGLCWLVSFLVGLTPMFGWNMKLTSEYHRNVTFLSCQFVSVMRMDYMVYFSFLTWIFIPLVVMCAIYLDIFYIIRNKLSLNLSNSKETGAFYGREFKTAKSLFLVLFLFALSWLPLSIINCIIYFNGEVPQLVLYMGILLSHANSMMNPIVYAYKIKKFKETYLLILKACVVCHPSDSLDTSIEKNSE