Reaction Details Report a problem with these data
Target
Cysteinyl leukotriene receptor 1
Ligand
BDBM50006798
Substrate
n/a
Meas. Tech.
ChEMBL_52044 (CHEMBL884353)
IC50
23±n/a nM
Citation
 Shaw, A; Krell, RD Peptide leukotrienes: current status of research. J Med Chem 34:1235-42 (1991) [PubMed]  Article 
Target
Name:
Cysteinyl leukotriene receptor 1
Synonyms:
CLTR1_CAVPO | CYSLTR1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
39007.58
Organism:
GUINEA PIG
Description:
Leukotriene D4 0 GUINEA PIG::Q2NNR5
Residue:
340
Sequence:
MDETGNPTIPPASNNTCYDSIDDFRNQVYSTLYSMISVVGFFGNGFVLYVLVKTYHEKSAFQVYMINLAVADLLCVCTLPLRVAYYVHKGIWLFGDFLCRLSTYALYVNLYCSIFFMTAMSFFRCVAIVFPVQNISLVTQKKARLVCIAIWMFVILTSSPFLMANTYKDEKNNTKCFEPPQDNQAKNYVLILHYVSLFIGFIIPFITIIVCYTMIIFTLLKSSMKKNLSSRKRAIGMIIVVTAAFLVSFMPYHIQRTIHLHFLHNKTKPCDSILRMQKSVVITLSLAASNCCFDPLLYFFSGGNFRRRLSTIRKYSLSSMTYIPKKKTSLPQKGKDICKE
  
Inhibitor
Name:
BDBM50006798
Synonyms:
2-[3-(Quinolin-2-ylmethoxy)-phenylamino]-benzoic acid | 2-[3-(Quinolin-2-ylmethoxy)-phenylamino]-benzoic acid(SR2640) | CHEMBL18132 | cid_128355
Type:
Small organic molecule
Emp. Form.:
C23H18N2O3
Mol. Mass.:
370.4006
SMILES:
OC(=O)c1ccccc1Nc1cccc(OCc2ccc3ccccc3n2)c1
Structure:
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