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Target
Adenosine receptor A2b
Ligand
BDBM50478191
Substrate
n/a
Meas. Tech.
ChEMBL_471614 (CHEMBL941043)
Ki
13±n/a nM
Citation
 Martínez, A; Gutiérrez-de-Terán, H; Brea, J; Raviña, E; Loza, MI; Cadavid, MI; Sanz, F; Vidal, B; Segarra, V; Sotelo, E Synthesis, adenosine receptor binding and 3D-QSAR of 4-substituted 2-(2'-furyl)-1,2,4-triazolo[1,5-a]quinoxalines. Bioorg Med Chem 16:2103-13 (2008) [PubMed]  Article 
Target
Name:
Adenosine receptor A2b
Synonyms:
AA2BR_HUMAN | ADENOSINE A2B | ADORA2B | Adenosine receptor A2B (A2B) | Adenosine receptors A2b | Adenosine receptors; A2a & A2b
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
36341.22
Organism:
Homo sapiens (Human)
Description:
n/a
Residue:
332
Sequence:
MLLETQDALYVALELVIAALSVAGNVLVCAAVGTANTLQTPTNYFLVSLAAADVAVGLFAIPFAITISLGFCTDFYGCLFLACFVLVLTQSSIFSLLAVAVDRYLAICVPLRYKSLVTGTRARGVIAVLWVLAFGIGLTPFLGWNSKDSATNNCTEPWDGTTNESCCLVKCLFENVVPMSYMVYFNFFGCVLPPLLIMLVIYIKIFLVACRQLQRTELMDHSRTTLQREIHAAKSLAMIVGIFALCWLPVHAVNCVTLFQPAQGKNKPKWAMNMAILLSHANSVVNPIVYAYRNRDFRYTFHKIISRYLLCQADVKSGNGQAGVQPALGVGL
  
Inhibitor
Name:
BDBM50478191
Synonyms:
CHEMBL261345
Type:
Small organic molecule
Emp. Form.:
C13H9N5O
Mol. Mass.:
251.2435
SMILES:
Nc1nc2ccccc2n2nc(nc12)-c1ccco1
Structure:
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