Reaction Details Report a problem with these data
Target
COP9 signalosome complex subunit 5
Ligand
BDBM50514114
Substrate
n/a
Meas. Tech.
ChEMBL_1855690 (CHEMBL4356419)
IC50
5.8±n/a nM
Citation
Schauer, NJ; Magin, RS; Liu, X; Doherty, LM; Buhrlage, SJ Advances in Discovering Deubiquitinating Enzyme (DUB) Inhibitors. J Med Chem 63:2731-2750 (2020) [PubMed] Article
More Info.:
Target
Name:
COP9 signalosome complex subunit 5
Synonyms:
COP9 signalosome complex subunit 5 (Csn5) | COPS5 | CSN5 | CSN5_HUMAN | JAB1
Type:
Protein
Mol. Mass.:
37578.39
Organism:
Homo sapiens (Human)
Description:
Q92905
Residue:
334
Sequence:
MAASGSGMAQKTWELANNMQEAQSIDEIYKYDKKQQQEILAAKPWTKDHHYFKYCKISALALLKMVMHARSGGNLEVMGLMLGKVDGETMIIMDSFALPVEGTETRVNAQAAAYEYMAAYIENAKQVGRLENAIGWYHSHPGYGCWLSGIDVSTQMLNQQFQEPFVAVVIDPTRTISAGKVNLGAFRTYPKGYKPPDEGPSEYQTIPLNKIEDFGVHCKQYYALEVSYFKSSLDRKLLELLWNKYWVNTLSSSSLLTNADYTTGQVFDLSEKLEQSEAQLGRGSFMLGLETHDRKSEDKLAKATRDSCKTTIEAIHGLMSQVIKDKLFNQINIS