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Target
Mu-type opioid receptor
Ligand
BDBM50070947
Substrate
n/a
Meas. Tech.
ChEBML_138741
Ki
102±n/a nM
Citation
 Tsai, YC; Liou, JP; Liao, R; Cheng, CY; Tao, PL C-alkylated spiro[benzofuran-3(2H),4'-1'-methyl-piperidine-7-ols] as potent opioids: a conformation-activity study. Bioorg Med Chem Lett 8:1813-8 (1999) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50070947
Synonyms:
2-ethyl-1'-methylspiro[2,3-dihydrobenzo[b]furan-3,4'-(hexahydropyridine)]-7-ol | CHEMBL431156
Type:
Small organic molecule
Emp. Form.:
C15H21NO2
Mol. Mass.:
247.3327
SMILES:
CCC1Oc2c(cccc2O)C11CCN(C)CC1
Structure:
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