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Target
Probable G-protein coupled receptor 34
Ligand
BDBM50560836
Substrate
n/a
Meas. Tech.
ChEMBL_2073602 (CHEMBL4729136)
EC50
>3000±n/a nM
Citation
 Nakamura, S; Sayama, M; Uwamizu, A; Jung, S; Ikubo, M; Otani, Y; Kano, K; Omi, J; Inoue, A; Aoki, J; Ohwada, T Non-naturally Occurring Regio Isomer of Lysophosphatidylserine Exhibits Potent Agonistic Activity toward G Protein-Coupled Receptors. J Med Chem 63:9990-10029 (2020) [PubMed]  Article 
Target
Name:
Probable G-protein coupled receptor 34
Synonyms:
gpr34a
Type:
PROTEIN
Mol. Mass.:
44073.38
Organism:
Danio rerio
Description:
ChEMBL_120175
Residue:
389
Sequence:
MSSTESLQSFSSVWDNRSMWSNRSCPLEEEALRLPLAVLYSLIFLFGLLGNLLALWVFLFLHRRRNSVRVFLINVALADLVLLACLPFRVLYHALGNVWTLGPRMCRVVGNLFYMNMYVSITLLGLISLDRYLKIMGSHRGRRWLRGRSWSLVTCGLLWGLSVLMAVPMMALAEGNEEPGKCYQYKQRKHARGKAYFNLVMVAVFWLVFVVLLVSYGQIARRLLRASQDKPHLPNAARYARTARKSFVVPLLFTVCFVPYHAFRGFYVASQLQDISCETRRLMDRTNEAVLLLSALNSCLDPVMYFLLSGSVRRATLQALAQCLRLHAEPPATNSSTTELRRTSVSHASTTAVLDTSRCSLGNITTLRSQHTDLHPHSEPCVHRSGLSD
  
Inhibitor
Name:
BDBM50560836
Synonyms:
CHEMBL4758243
Type:
Small organic molecule
Emp. Form.:
C30H36NO11P
Mol. Mass.:
617.5807
SMILES:
CCOC[C@H](COC(=O)CCc1ccccc1OCc1cccc(Oc2ccccc2)c1)OP(O)(=O)OC[C@H](N)C(O)=O |r|
Structure:
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