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Target
Testis-specific serine/threonine-protein kinase 2
Ligand
BDBM50582077
Substrate
n/a
Meas. Tech.
ChEMBL_2153006 (CHEMBL5037553)
IC50
944±n/a nM
Citation
Elsner, J; Cashion, D; Robinson, D; Bahmanyar, S; Tehrani, L; Fultz, KE; Narla, RK; Peng, X; Tran, T; Apuy, J; LeBrun, L; Leftheris, K; Boylan, JF; Zhu, D; Riggs, JR Structure-Guided Optimization Provides a Series of TTK Protein Inhibitors with Potent Antitumor Activity. J Med Chem 64:12670-12679 (2021) [PubMed] Article
More Info.:
Target
Name:
Testis-specific serine/threonine-protein kinase 2
Synonyms:
DGSG | SPOGA2 | STK22B | TSSK2 | TSSK2_HUMAN
Type:
PROTEIN
Mol. Mass.:
40954.93
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1459845
Residue:
358
Sequence:
MDDATVLRKKGYIVGINLGKGSYAKVKSAYSERLKFNVAVKIIDRKKTPTDFVERFLPREMDILATVNHGSIIKTYEIFETSDGRIYIIMELGVQGDLLEFIKCQGALHEDVARKMFRQLSSAVKYCHDLDIVHRDLKCENLLLDKDFNIKLSDFGFSKRCLRDSNGRIILSKTFCGSAAYAAPEVLQSIPYQPKVYDIWSLGVILYIMVCGSMPYDDSDIRKMLRIQKEHRVDFPRSKNLTCECKDLIYRMLQPDVSQRLHIDEILSHSWLQPPKPKATSSASFKREGEGKYRAECKLDTKTGLRPDHRPDHKLGAKTQHRLLVVPENENRMEDRLAETSRAKDHHISGAEVGKAST