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Target
D(3) dopamine receptor
Ligand
BDBM50596494
Substrate
n/a
Meas. Tech.
ChEMBL_2220553 (CHEMBL5133887)
Ki
52±n/a nM
Citation
 Elek, M; Dubiel, M; Mayer, L; Zivkovic, A; Müller, TJJ; Stark, H BOPPY-based novel fluorescent dopamine D Bioorg Med Chem Lett 59:0 (2022) [PubMed] 
Target
Name:
D(3) dopamine receptor
Synonyms:
DRD3 | DRD3_HUMAN | Dopamine D3 receptor
Type:
PROTEIN
Mol. Mass.:
44213.40
Organism:
Homo sapiens
Description:
ChEMBL_105671
Residue:
400
Sequence:
MASLSQLSGHLNYTCGAENSTGASQARPHAYYALSYCALILAIVFGNGLVCMAVLKERALQTTTNYLVVSLAVADLLVATLVMPWVVYLEVTGGVWNFSRICCDVFVTLDVMMCTASILNLCAISIDRYTAVVMPVHYQHGTGQSSCRRVALMITAVWVLAFAVSCPLLFGFNTTGDPTVCSISNPDFVIYSSVVSFYLPFGVTVLVYARIYVVLKQRRRKRILTRQNSQCNSVRPGFPQQTLSPDPAHLELKRYYSICQDTALGGPGFQERGGELKREEKTRNSLSPTIAPKLSLEVRKLSNGRLSTSLKLGPLQPRGVPLREKKATQMVAIVLGAFIVCWLPFFLTHVLNTHCQTCHVSPELYSATTWLGYVNSALNPVIYTTFNIEFRKAFLKILSC
  
Inhibitor
Name:
BDBM50596494
Synonyms:
CHEMBL5207676
Type:
Small organic molecule
Emp. Form.:
C28H35B2Cl2F4N7
Mol. Mass.:
638.146
SMILES:
CCc1c(C)c2C=[N+]3[N+](=C4C=CC=C(NCCCCN5CCN(CC5)c5cccc(Cl)c5Cl)N4[B-]3(F)F)[B-](F)(F)n2c1C |c:6,10,t:8,12|
Structure:
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