Reaction Details Report a problem with these data
Target
Malate dehydrogenase
Ligand
BDBM50023867
Substrate
n/a
Meas. Tech.
ChEMBL_103875 (CHEMBL712992)
IC50
30000±n/a nM
Citation
McGovern, SL; Shoichet, BK Kinase inhibitors: not just for kinases anymore. J Med Chem 46:1478-83 (2003) [PubMed] Article
More Info.:
Target
Name:
Malate dehydrogenase
Synonyms:
MDH_THETH | mdh
Type:
PROTEIN
Mol. Mass.:
35423.44
Organism:
Thermus thermophilus
Description:
ChEMBL_1448377
Residue:
327
Sequence:
MKAPVRVAVTGAAGQIGYSLLFRIAAGEMLGKDQPVILQLLEIPQAMKALEGVVMELEDCAFPLLAGLEATDDPKVAFKDADYALLVGAAPRKAGMERRDLLQVNGKIFTEQGRALAEVAKKDVKVLVVGNPANTNALIAYKNAPGLNPRNFTAMTRLDHNRAKAQLAKKTGTGVDRIRRMTVWGNHSSTMFPDLFHAEVDGRPALELVDMEWYEKVFIPTVAQRGAAIIQARGASSAASAANAAIEHIRDWALGTPEGDWVSMAVPSQGEYGIPEGIVYSFPVTAKDGAYRVVEGLEINEFARKRMEITAQELLDEMEQVKALGLI