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Target
DNA-directed DNA/RNA polymerase mu
Ligand
BDBM50379292
Substrate
n/a
Meas. Tech.
ChEMBL_811412 (CHEMBL2013670)
IC50
>200000±n/a nM
Citation
Myobatake, Y; Takeuchi, T; Kuramochi, K; Kuriyama, I; Ishido, T; Hirano, K; Sugawara, F; Yoshida, H; Mizushina, Y Pinophilins A and B, inhibitors of mammalian A-, B-, and Y-family DNA polymerases and human cancer cell proliferation. J Nat Prod 75:135-41 (2012) [PubMed] Article
More Info.:
Target
Name:
DNA-directed DNA/RNA polymerase mu
Synonyms:
DPOLM_HUMAN | POLM | Pol Mu | Terminal transferase | polmu
Type:
PROTEIN
Mol. Mass.:
54829.49
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1297319
Residue:
494
Sequence:
MLPKRRRARVGSPSGDAASSTPPSTRFPGVAIYLVEPRMGRSRRAFLTGLARSKGFRVLDACSSEATHVVMEETSAEEAVSWQERRMAAAPPGCTPPALLDISWLTESLGAGQPVPVECRHRLEVAGPRKGPLSPAWMPAYACQRPTPLTHHNTGLSEALEILAEAAGFEGSEGRLLTFCRAASVLKALPSPVTTLSQLQGLPHFGEHSSRVVQELLEHGVCEEVERVRRSERYQTMKLFTQIFGVGVKTADRWYREGLRTLDDLREQPQKLTQQQKAGLQHHQDLSTPVLRSDVDALQQVVEEAVGQALPGATVTLTGGFRRGKLQGHDVDFLITHPKEGQEAGLLPRVMCRLQDQGLILYHQHQHSCCESPTRLAQQSHMDAFERSFCIFRLPQPPGAAVGGSTRPCPSWKAVRVDLVVAPVSQFPFALLGWTGSKLFQRELRRFSRKEKGLWLNSHGLFDPEQKTFFQAASEEDIFRHLGLEYLPPEQRNA