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Target
Serine racemase
Ligand
BDBM50444848
Substrate
n/a
Meas. Tech.
ChEMBL_1282560 (CHEMBL3101227)
Ki
661000000±n/a nM
Citation
 Harty, M; Nagar, M; Atkinson, L; Legay, CM; Derksen, DJ; Bearne, SL Inhibition of serine and proline racemases by substrate-product analogues. Bioorg Med Chem Lett 24:390-3 (2013) [PubMed]  Article 
Target
Name:
Serine racemase
Synonyms:
D-serine ammonia-lyase | D-serine dehydratase | L-serine ammonia-lyase | L-serine dehydratase | SPCC330.15c | SRR | SRR_SCHPO
Type:
PROTEIN
Mol. Mass.:
35050.33
Organism:
Schizosaccharomyces pombe (strain 972 / ATCC 24843) (Fission yeast)
Description:
ChEMBL_107985
Residue:
323
Sequence:
MSDNLVLPTYDDVASASERIKKFANKTPVLTSSTVNKEFVAEVFFKCENFQKMGAFKFRGALNALSQLNEAQRKAGVLTFSSGNHAQAIALSAKILGIPAKIIMPLDAPEAKVAATKGYGGQVIMYDRYKDDREKMAKEISEREGLTIIPPYDHPHVLAGQGTAAKELFEEVGPLDALFVCLGGGGLLSGSALAARHFAPNCEVYGVEPEAGNDGQQSFRKGSIVHIDTPKTIADGAQTQHLGNYTFSIIKEKVDDILTVSDEELIDCLKFYAARMKIVVEPTGCLSFAAARAMKEKLKNKRIGIIISGGNVDIERYAHFLSQ
  
Inhibitor
Name:
BDBM50444848
Synonyms:
CHEMBL3099359
Type:
Small organic molecule
Emp. Form.:
C4H9NO4
Mol. Mass.:
135.1186
SMILES:
[NH3+]C(CO)(CO)C([O-])=O
Structure:
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