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Target
Solute carrier organic anion transporter family member 2B1
Ligand
BDBM50101853
Substrate
n/a
Meas. Tech.
ChEMBL_836786 (CHEMBL2075311)
IC50
36±n/a nM
Citation
 Nishio, T; Adachi, H; Nakagomi, R; Tokui, T; Sato, E; Tanemoto, M; Fujiwara, K; Okabe, M; Onogawa, T; Suzuki, T; Nakai, D; Shiiba, K; Suzuki, M; Ohtani, H; Kondo, Y; Unno, M; Ito, S; Iinuma, K; Nunoki, K; Matsuno, S; Abe, T Molecular identification of a rat novel organic anion transporter moat1, which transports prostaglandin D(2), leukotriene C(4), and taurocholate. Biochem Biophys Res Commun 275:831-8 (2000) [PubMed]  Article 
Target
Name:
Solute carrier organic anion transporter family member 2B1
Synonyms:
Organic anion transporter moatp1 | Solute carrier family 21 member 9 | SO2B1_RAT | Slco2b1 | Oatp2b1 | Slc21a9
Type:
PROTEIN
Mol. Mass.:
74232.20
Organism:
Rat
Description:
ChEMBL_104639
Residue:
682
Sequence:
MPDRSTKATMGAEDIHERKVSMEPRDSHQDAQPRGMFQNIKFFVLCHSILQLAQLMISGYLKSSISTVEKRFGLSSQTSGLLAAFNEVGNISLILFVSYFGSRVHRPRMIGCGAILVAVAGLLMALPHFISEPYRYDHSSPDRSQDFEASLCLPTTMAPASALSNDSCSSRTETKHLTMVGIMFTAQTLLGIGGVPIQPFGISYIDDFAHHSNSPLYLGILFAITMMGPGLAYGLGSLMLRLYVDIDRMPEGGINLTTKDPRWVGAWWLGFLISAGLVVLAASPYFFFPREMPKEKYELHFRQKVLAGGASIGSKGEELSSQHEPLKKQAGLPQIAPDLTVVQFIKVFPRVLLRTLRHPIFLLVVLSQVCTSSMVAGTATFLPKFLERQFSITASFANLLLGCLTIPLAIVGIVVGGVLVKRLHLSPMQCSALCLLGSLLCLLLSLPLFFIGCSTHHIAGITQDLGAQPGPSLFPGCSEPCSCQSDDFNPVCDTSAYVEYTTPCHAGCTGRVVQEALDKSQVFYTNCSCVAGNGTISAGSCESACSRLVLPFILLISLGAAVASITHTPSFMLILRGVKKEDKTLAVGMQFMLLRVLAWMPSPVIHGSAIDTTCVHWALTCGRRAVCRYYDHDLLRNRFIGLQFFFKSGSLVCFALVLAILRQQSREASTKATVKSSDLQEL
  
Inhibitor
Name:
BDBM50101853
Synonyms:
(13E,15S)-11alpha,15-dihydroxy-9-oxoprost-13-en-1-oic acid | prostaglandin E1 | (11alpha,13E,15S)-11,15-dihydroxy-9-oxoprost-13-en-1-oic acid | 11alpha,15alpha-dihydroxy-9-oxo-13-trans-prostenoic acid | PGE-1 | PGE1 | CHEMBL495 | ALPROSTADIL
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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