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Target
Delta-type opioid receptor
Ligand
BDBM50412268
Substrate
n/a
Meas. Tech.
ChEMBL_1462230 (CHEMBL3395162)
Ki
37500±n/a nM
Citation
 Ruiu, S; Anzani, N; Orrų, A; Floris, C; Caboni, P; Alcaro, S; Maccioni, E; Distinto, S; Cottiglia, F Methoxyflavones from Stachys glutinosa with binding affinity to opioid receptors: in silico, in vitro, and in vivo studies. J Nat Prod 78:69-76 (2015) [PubMed]  Article 
Target
Name:
Delta-type opioid receptor
Synonyms:
DOR-1 | K56 | MSL-2 | OPIATE Delta | OPRD_MOUSE | Opioid receptors; mu and delta | Oprd1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
40577.25
Organism:
MOUSE
Description:
P32300
Residue:
372
Sequence:
MELVPSARAELQSSPLVNLSDAFPSAFPSAGANASGSPGARSASSLALAIAITALYSAVCAVGLLGNVLVMFGIVRYTKLKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELLCKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVGVPIMVMAVTQPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRLRSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDINRRDPLVVAALHLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRTPCGRQEPGSLRRPRQATTRERVTACTPSDGPGGGAAA
  
Inhibitor
Name:
BDBM50412268
Synonyms:
CHEMBL74272
Type:
Small organic molecule
Emp. Form.:
C19H18O8
Mol. Mass.:
374.3414
SMILES:
COc1cc(ccc1O)-c1cc(=O)c2c(O)c(OC)c(OC)c(OC)c2o1
Structure:
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