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Target
Ribosomal protein S6 kinase alpha-3
Ligand
BDBM50111366
Substrate
n/a
Meas. Tech.
ChEMBL_1509948 (CHEMBL3607766)
EC50
6400±n/a nM
Citation
Jain, R; Mathur, M; Lan, J; Costales, A; Atallah, G; Ramurthy, S; Subramanian, S; Setti, L; Feucht, P; Warne, B; Doyle, L; Basham, S; Jefferson, AB; Lindvall, M; Appleton, BA; Shafer, CM Discovery of Potent and Selective RSK Inhibitors as Biological Probes. J Med Chem 58:6766-83 (2015) [PubMed] Article
More Info.:
Target
Name:
Ribosomal protein S6 kinase alpha-3
Synonyms:
90 kDa ribosomal protein S6 kinase 3 | KS6A3_MOUSE | MAP kinase-activated protein kinase 1b | MAPK-activated protein kinase 1b | MAPKAP kinase 1b | MAPKAPK-1b | Mapkapk1b | Mapkapk1b | RSK-2 | Ribosomal S6 kinase 2 | Ribosomal protein S6 kinase alpha-3 | Rps6ka-rs1 | Rps6ka3 | Rsk2 | S6K-alpha-3 | p90-RSK 3 | p90RSK3 | pp90RSK2
Type:
PROTEIN
Mol. Mass.:
83697.95
Organism:
Mus musculus
Description:
ChEMBL_108393
Residue:
740
Sequence:
MPLAQLADPWQKMAVESPSDSAENGQQIMDEPMGEEEINPQTEEGSIKEIAITHHVKEGHEKADPSQFELLKVLGQGSFGKVFLVKKISGSDARQLYAMKVLKKATLKVRDRVRTKMERDILVEVNHPFIVKLHYAFQTEGKLYLILDFLRGGDLFTRLSKEVMFTEEDVKFYLAELALALDHLHSLGIIYRDLKPENILLDEEGHIKLTDFGLSKESIDHEKKAYSFCGTVEYMAPEVVNRRGHTQSADWWSFGVLMFEMLTGTLPFQGKDRKETMTMILKAKLGMPQFLSPEAQSLLRMLFKRNPANRLGAGPDGVEEIKRHSFFSTIDWNKLYRREIHPPFKPATGRPEDTFYFDPEFTAKTPKDSPGIPPSANAHQLFRGFSFVAITSDDESQAMQTVGVHSIVQQLHRNSIQFTDGYEVKEDIGVGSYSVCKRCIHKATNMEFAVKIIDKSKRDPTEEIEILLRYGQHPNIITLKDVYDDGKYVYVVTELMKGGELLDKILRQKFFSEREASAVLFTITKTVEYLHAQGVVHRDLKPSNILYVDESGNPESIRICDFGFAKQLRAENGLLMTPCYTANFVAPEVLKRQGYDAACDIWSLGVLLYTMLTGYTPFANGPDDTPEEILARIGSGKFSLSGGYWNSVSDTAKDLVSKMLHVDPHQRLTAALVLRHPWIVHWDQLPQYQLNRQDAPHLVKGAMAATYSALNRNQSPVLEPVGRSTLAQRRGIKKITSTAL