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Target
Histamine receptor H4
Ligand
BDBM7966
Substrate
n/a
Ki
104±n/a nM
Comments
PDSP_934
Citation
Zhu, Y; Michalovich, D; Wu, H; Tan, KB; Dytko, GM; Mannan, IJ; Boyce, R; Alston, J; Tierney, LA; Li, X; Herrity, NC; Vawter, L; Sarau, HM; Ames, RS; Davenport, CM; Hieble, JP; Wilson, S; Bergsma, DJ; Fitzgerald, LR Cloning, expression, and pharmacological characterization of a novel human histamine receptor. Mol Pharmacol 59:434-41 (2001) [PubMed] Article
More Info.:
Target
Name:
Histamine receptor H4
Synonyms:
HISTAMINE H4 | HRH4 | Histamine H4 receptor
Type:
Enzyme Catalytic Domain
Mol. Mass.:
44536.99
Organism:
GUINEA PIG
Description:
HISTAMINE H4 HRH4 GUINEA PIG::Q91ZY3
Residue:
389
Sequence:
MLANNSTIALTSIKISLTFLMSLLAIAIMLGNVVVILAFIVDRNLRHRSNYFFLNLAIADFFVGAIAIPLYIPSSLTYWTSGKQACVFWLITDYLLCTASVYNIVLISYDRYQSVSNAVWYRAQHSGTWKIATQMVAVWIFSFMTNGPMILISDSWQNSTTECEPGFLKKWYFALPTSLLEFLIPILLVAYFSAHIYWSLWKREKLSRCLSHPVLPSDSSSSDHGHSCRQDPDSRATLPARKETTASLGSDKSRRKSSLLFSIRAYKNSNVIASKMGFLSHSDSLALQQREHIELFRARKLAKSLAILLAAFAICWAPYSLTTVIYSFFPERNLTKSTWYHTAFWLQWFNSFVNPFLYPLCHKRFQKAFLKILPVRRQSTPPHNRSIST