Reaction Details Report a problem with these data
Target
Cyclin-dependent kinase 16
Ligand
BDBM186184
Substrate
n/a
Meas. Tech.
LanthaScreen TR-FRET Assay
Temperature
295.15±n/a K
IC50
1.50e+3±n/a nM
Comments
extracted
Citation
Alisi, MA; Cazzolla, N; Garofalo, B; Furlotti, G; Magaro′, G; Ombrato, R; Mancini, F Use of 1H-indazole-3-carboxamide compounds as glycogen synthase kinase 3 beta inhibitors US Patent US9163013 Publication Date 10/20/2015
More Info.:
Target
Name:
Cyclin-dependent kinase 16
Synonyms:
CDK16 | CDK16_HUMAN | PCTAIRE1 | PCTK1 | Serine/threonine-protein kinase PCTAIRE-1
Type:
Protein
Mol. Mass.:
55721.58
Organism:
Homo sapiens (Human)
Description:
Q00536
Residue:
496
Sequence:
MDRMKKIKRQLSMTLRGGRGIDKTNGAPEQIGLDESGGGGGSDPGEAPTRAAPGELRSARGPLSSAPEIVHEDLKMGSDGESDQASATSSDEVQSPVRVRMRNHPPRKISTEDINKRLSLPADIRLPEGYLEKLTLNSPIFDKPLSRRLRRVSLSEIGFGKLETYIKLDKLGEGTYATVYKGKSKLTDNLVALKEIRLEHEEGAPCTAIREVSLLKDLKHANIVTLHDIIHTEKSLTLVFEYLDKDLKQYLDDCGNIINMHNVKLFLFQLLRGLAYCHRQKVLHRDLKPQNLLINERGELKLADFGLARAKSIPTKTYSNEVVTLWYRPPDILLGSTDYSTQIDMWGVGCIFYEMATGRPLFPGSTVEEQLHFIFRILGTPTEETWPGILSNEEFKTYNYPKYRAEALLSHAPRLDSDGADLLTKLLQFEGRNRISAEDAMKHPFFLSLGERIHKLPDTTSIFALKEIQLQKEASLRSSSMPDSGRPAFRVVDTEF