Reaction Details Report a problem with these data
Target
Fatty acid-binding protein, adipocyte
Ligand
BDBM50429939
Substrate
n/a
Meas. Tech.
Fluorescent Displacement Assay
IC50
1100±n/a nM
Citation
 Fukunaga, K; Miyachi, H; Ishida, H; Ban, S Agent for treating synucleinopathy US Patent  US10709688 Publication Date 7/14/2020 
Target
Name:
Fatty acid-binding protein, adipocyte
Synonyms:
A-FABP | AFABP | ALBP | Adipocyte lipid-binding protein | FABP4 | FABP4_HUMAN | Fatty acid binding protein adipocyte | Fatty acid-binding protein 4 | Fatty acid-binding protein 4 (FABP4)
Type:
Enzyme
Mol. Mass.:
14719.23
Organism:
Homo sapiens (Human)
Description:
P15090
Residue:
132
Sequence:
MCDAFVGTWKLVSSENFDDYMKEVGVGFATRKVAGMAKPNMIISVNGDVITIKSESTFKNTEISFILGQEFDEVTADDRKVKSTITLDGGVLVHVQKWDGKSTTIKRKREDDKLVVECVMKGVTSTRVYERA
  
Inhibitor
Name:
BDBM50429939
Synonyms:
CHEMBL2334261 | US10709688, Example 6
Type:
Small organic molecule
Emp. Form.:
C25H21ClN2O3
Mol. Mass.:
432.899
SMILES:
OC(=O)CCCOc1ccccc1-c1cc(-c2ccccc2)n(n1)-c1cccc(Cl)c1
Structure:
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