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Found 456 with Last Name = 'ishida' and Initial = 'h'
TargetSialidase-2(Homo sapiens (Human))
Gifu University

Curated by ChEMBL
LigandPNGBDBM50295841(4-Acetamido-5-(biphenyl-4-ylcarboxamido)-2-fluorob...)
Affinity DataKi:  3.07E+5nMAssay Description:Inhibition of human NEU2 transiently transfected in HEK293 cells by Line-Weaver Burk plottingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Bos taurus)
Ochanomizu University

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataIC50:  0.0480nMAssay Description:Displacement of [3H]-1-alpha,25-(OH)2D3 from bovine thymus VDR incubated for 18 hrs by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Showa Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataIC50:  0.160nMAssay Description:Displacement of [3H]-1,25-(OH)2D3 from N-terminal GST-tagged human recombinant vitamin D receptor ligand binding domain expressed in Escherichia coli...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391561(CHEMBL2147704)
Affinity DataIC50:  0.180nMAssay Description:Inhibition of DPP4 in rat plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391559(CHEMBL2147703)
Affinity DataIC50:  0.190nMAssay Description:Inhibition of DPP4 in rat plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391561(CHEMBL2147704)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of DPP4 in human plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391559(CHEMBL2147703)
Affinity DataIC50:  0.260nMAssay Description:Inhibition of DPP4 in human plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391565(CHEMBL2147777)
Affinity DataIC50:  0.290nMAssay Description:Inhibition of DPP4 in rat plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391570(CHEMBL2147712)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of DPP4 in human plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391567(CHEMBL2147709)
Affinity DataIC50:  0.310nMAssay Description:Inhibition of DPP4 in rat plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391567(CHEMBL2147709)
Affinity DataIC50:  0.320nMAssay Description:Inhibition of DPP4 in human plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Thammasat University

Curated by ChEMBL
LigandPNGBDBM50182249(CHEMBL3818159)
Affinity DataIC50:  0.350nMAssay Description:Inhibition of Influenza A virus (A/duck/Tsukuba/28/2005(H6N2)) neuraminidase N2 activity using 4MU-Neu5Ac as substrate preincubated for 15 mins follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391565(CHEMBL2147777)
Affinity DataIC50:  0.370nMAssay Description:Inhibition of DPP4 in human plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388112(CHEMBL2058971)
Affinity DataIC50:  0.370nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388112(CHEMBL2058971)
Affinity DataIC50:  0.370nMAssay Description:Inhibition of DPP4 in human plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388123(CHEMBL2058762)
Affinity DataIC50:  0.390nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388127(CHEMBL2058758)
Affinity DataIC50:  0.420nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Thammasat University

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50:  0.470nMAssay Description:Inhibition of Influenza A virus (A/duck/Tsukuba/67/2005(H1N1)) neuraminidase N1 activity using 4MU-Neu5Ac as substrate preincubated for 15 mins follo...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391570(CHEMBL2147712)
Affinity DataIC50:  0.490nMAssay Description:Inhibition of DPP4 in rat plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388125(CHEMBL2058756)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388115(CHEMBL2058975)
Affinity DataIC50:  0.510nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Thammasat University

Curated by ChEMBL
LigandPNGBDBM50182249(CHEMBL3818159)
Affinity DataIC50:  0.530nMAssay Description:Inhibition of Influenza A virus (A/duck/Tsukuba/394/2005(H5N3)) neuraminidase N3 activity using 4MU-Neu5Ac as substrate preincubated for 15 mins foll...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391571(CHEMBL2147713)
Affinity DataIC50:  0.530nMAssay Description:Inhibition of DPP4 in rat plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388126(CHEMBL2058757)
Affinity DataIC50:  0.550nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388118(CHEMBL2058970)
Affinity DataIC50:  0.560nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388115(CHEMBL2058975)
Affinity DataIC50:  0.560nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Thammasat University

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50:  0.580nMAssay Description:Inhibition of Influenza A virus (A/duck/Tsukuba/20/2007(H8N4)) neuraminidase N4 activity using 4MU-Neu5Ac as substrate preincubated for 15 mins follo...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388112(CHEMBL2058971)
Affinity DataIC50:  0.590nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388122(CHEMBL2058761)
Affinity DataIC50:  0.590nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388113(CHEMBL2058973)
Affinity DataIC50:  0.610nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388119(CHEMBL2058972)
Affinity DataIC50:  0.610nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388123(CHEMBL2058762)
Affinity DataIC50:  0.610nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388119(CHEMBL2058972)
Affinity DataIC50:  0.620nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391576(CHEMBL2147773)
Affinity DataIC50:  0.620nMAssay Description:Inhibition of DPP4 in human plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391568(CHEMBL2147771)
Affinity DataIC50:  0.630nMAssay Description:Inhibition of DPP4 in human plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388127(CHEMBL2058758)
Affinity DataIC50:  0.690nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391564(CHEMBL2147707)
Affinity DataIC50:  0.690nMAssay Description:Inhibition of DPP4 in rat plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388125(CHEMBL2058756)
Affinity DataIC50:  0.720nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391568(CHEMBL2147771)
Affinity DataIC50:  0.720nMAssay Description:Inhibition of DPP4 in rat plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388114(CHEMBL2058974)
Affinity DataIC50:  0.730nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388126(CHEMBL2058757)
Affinity DataIC50:  0.770nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391576(CHEMBL2147773)
Affinity DataIC50:  0.770nMAssay Description:Inhibition of DPP4 in rat plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388114(CHEMBL2058974)
Affinity DataIC50:  0.790nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388121(CHEMBL2058760)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus)
Thammasat University

Curated by ChEMBL
LigandPNGBDBM50182249(CHEMBL3818159)
Affinity DataIC50:  0.810nMAssay Description:Inhibition of Influenza A virus (A/duck/Tsukuba/700/2007(H7N7)) neuraminidase N7 activity using 4MU-Neu5Ac as substrate preincubated for 15 mins foll...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Rattus norvegicus (rat))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388113(CHEMBL2058973)
Affinity DataIC50:  0.830nMAssay Description:Inhibition of rat DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391571(CHEMBL2147713)
Affinity DataIC50:  0.850nMAssay Description:Inhibition of DPP4 in human plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50206043(((2S,4S)-4-(4-(5-nitropyridin-2-yl)piperazin-1-yl)...)
Affinity DataIC50:  0.920nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50391564(CHEMBL2147707)
Affinity DataIC50:  0.940nMAssay Description:Inhibition of DPP4 in human plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50388117(CHEMBL2058969)
Affinity DataIC50:  0.950nMAssay Description:Inhibition of DPP4 in human plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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