Report error Found 4 Enz. Inhib. hit(s) for PDB: 4CKR
TargetEpithelial discoidin domain-containing receptor 1(Human)
Massachusetts General Hospital and Harvard Medical School
Massachusetts General Hospital and Harvard Medical School
Affinity DataEC50: 86nMAssay Description:The enzyme kinase assay was carried out using the Lanthascreen technology.More data for this Ligand-Target Pair
3D Structure (crystal)TargetEpithelial discoidin domain-containing receptor 1(Human)
Massachusetts General Hospital and Harvard Medical School
Massachusetts General Hospital and Harvard Medical School
Affinity DataIC50: 86nMAssay Description:Inhibition of human DDR1 in doxycycline-stimulated human U2OS cells assessed as inhibition of collagen-1-induced autophosphorylation incubated for 1 ...More data for this Ligand-Target Pair
TargetEpithelial discoidin domain-containing receptor 1(Human)
Massachusetts General Hospital and Harvard Medical School
Massachusetts General Hospital and Harvard Medical School
Affinity DataIC50: 105nMAssay Description:Inhibition of human DDR1 kinase domain (601 to 913 residues) expressed in Sf9 cells by enzymatic kinase assayMore data for this Ligand-Target Pair
TargetEpithelial discoidin domain-containing receptor 1(Human)
Massachusetts General Hospital and Harvard Medical School
Massachusetts General Hospital and Harvard Medical School
Affinity DataIC50: 105nMAssay Description:Tet inducible human DDR1 over-expressing U2OS was pre-treated by media containing each of the compound for 1 hour and treated by changing the media t...More data for this Ligand-Target Pair