Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 5NLK
TargetCREB-binding protein(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50459793(CHEMBL4205572)
Affinity DataIC50: 19nMAssay Description:Displacement of biotinylated acetylated peptide from poly His-tagged CBP bromodomain (unknown origin) expressed in Escherichia coli BL21(DE3) by Alph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCREB-binding protein(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50459793(CHEMBL4205572)
Affinity DataKd:  35nMAssay Description:Binding affinity to Poly-Histidine-tagged CBP (unknown origin) expressed in Escherichia coli BL21(DE3) by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCREB-binding protein(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50459793(CHEMBL4205572)
Affinity DataKd:  35nMAssay Description:Displacement of biotinylated acetylated peptide from poly His-tagged CBP bromodomain (unknown origin) expressed in Escherichia coli BL21(DE3) measure...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)