Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) for PDB: 6DF7
LigandPNGBDBM50503406(CHEMBL4463538)
Affinity DataKd:  5nMAssay Description:Binding affinity to recombinant human full length DNA-tagged TAF1L bromodomain 2 (1523 to 1654 residues) expressed in bacterial expression system by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTranscription initiation factor TFIID subunit 1(Human)
Moffitt Cancer Center

Curated by ChEMBL
LigandPNGBDBM50503406(CHEMBL4463538)
Affinity DataKd:  39nMAssay Description:Binding affinity to human TAF1 tandem bromodomain (1373 to 1499 residues) transfected in Escherichia coli BL21 (DE3) assessed as dissociation constan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTranscription initiation factor TFIID subunit 1(Human)
Moffitt Cancer Center

Curated by ChEMBL
LigandPNGBDBM50503406(CHEMBL4463538)
Affinity DataEC50:  920nMAssay Description:Binding affinity to TAF1 in HEK293T cells assessed as increase in TAF1 level by ITDR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTranscription initiation factor TFIID subunit 1(Human)
Moffitt Cancer Center

Curated by ChEMBL
LigandPNGBDBM50503406(CHEMBL4463538)
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant His-tagged TAF1 bromodomain 2 (unknown origin) after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTranscription initiation factor TFIID subunit 1(Human)
Moffitt Cancer Center

Curated by ChEMBL
LigandPNGBDBM50503406(CHEMBL4463538)
Affinity DataIC50: 38nMAssay Description:Inhibition of fluorescent-tagged ligand from nanoLuc fused N-terminal TAF1 bromodomain 2 (unknown origin) expressed in 293T cells by luciferase repor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTranscription initiation factor TFIID subunit 1(Human)
Moffitt Cancer Center

Curated by ChEMBL
LigandPNGBDBM50503406(CHEMBL4463538)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of recombinant His-tagged TAF1 bromodomain 1 (unknown origin) after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)