Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) for PDB: 6JOE
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50519349(CHEMBL2431997)
Affinity DataKd:  91nMAssay Description:Binding affinity to Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50519349(CHEMBL2431997)
Affinity DataIC50: 180nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50519349(CHEMBL2431997)
Affinity DataIC50: 330nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 Rosetta (DE3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50519349(CHEMBL2431997)
Affinity DataIC50: 840nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 Rosetta (DE3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)