Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 6MXY
TargetTP53-binding protein 1(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM154565(N-(3-(Tert-butylamino)propyl)-3-(trifluoromethyl)b...)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of 53BP1 methyllysine binding domain (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTP53-binding protein 1(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM154565(N-(3-(Tert-butylamino)propyl)-3-(trifluoromethyl)b...)
Affinity DataIC50: 2.20E+4nMpH: 8.0 T: 2°CAssay Description:In brief, compound plates (1 μL at 10 mM highest concentration; 3-fold, 10-point dilutions in DMSO) were diluted in 1X assay buffer (20 mM TRIS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2015
Entry Details Article
PubMedPDB3D3D Structure (crystal)