Compile Data Set for Download or QSAR
Report error Found 132 of affinity data for UniProtKB/TrEMBL: O09778
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 29589BDBM29589(Panobinostat | Faridak | LBH-589B | LBH-589 | US10...)
Affinity DataEC50:  130nMAssay Description:Activation of Tat-mediated HIV1 transcription in J-Lat 10.6 cells harboring LTR driven GFP reporter co-expressing CMV driven RFP reporter assessed as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50048864BDBM50048864(CHEMBL3310505)
Affinity DataEC50:  220nMAssay Description:Activation of Tat-mediated HIV1 transcription in J-Lat 10.6 cells harboring LTR driven GFP reporter co-expressing CMV driven RFP reporter assessed as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524891BDBM50524891(CHEMBL4526214)
Affinity DataEC50:  800nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524887BDBM50524887(CHEMBL4446565)
Affinity DataEC50:  900nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50481913BDBM50481913(CHEMBL1075826)
Affinity DataIC50: 900nMAssay Description:Inhibition of HIV1 TAT transfected to human HeLa cells assessed as decrease in luminescence after 48 hrs by duel luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50476285BDBM50476285(CHEMBL609729)
Affinity DataEC50:  1.00E+3nMAssay Description:Inhibition of Tat-mediated transcription of viral promoter in 293 T cells transfected with HIV1 tat by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524928BDBM50524928(CHEMBL4457218)
Affinity DataEC50:  1.20E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524932BDBM50524932(CHEMBL4439301)
Affinity DataEC50:  1.30E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524948BDBM50524948(CHEMBL4450433)
Affinity DataEC50:  1.30E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524947BDBM50524947(CHEMBL4531178)
Affinity DataEC50:  1.40E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524929BDBM50524929(CHEMBL4582511)
Affinity DataEC50:  1.50E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524940BDBM50524940(CHEMBL4437258)
Affinity DataEC50:  1.70E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50410416BDBM50410416(CHEMBL196072)
Affinity DataKd:  1.80E+3nMT: 2°CAssay Description:In vitro binding affinity towards Tat/TAR to determine interaction between TAR RNA and Tat peptide at room temperature using fluorescence spectrophot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524889BDBM50524889(CHEMBL4552693)
Affinity DataEC50:  1.90E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524888BDBM50524888(CHEMBL4540359)
Affinity DataEC50:  2.20E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 19149BDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataEC50:  2.30E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in J-Lat 10.6 cells harboring LTR driven GFP reporter co-expressing CMV driven RFP reporter assessed as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524918BDBM50524918(CHEMBL4463956)
Affinity DataEC50:  2.30E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524930BDBM50524930(CHEMBL4555472)
Affinity DataEC50:  2.60E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524934BDBM50524934(CHEMBL4465487)
Affinity DataEC50:  2.60E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524945BDBM50524945(CHEMBL4464874)
Affinity DataEC50:  2.70E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524935BDBM50524935(CHEMBL4450555)
Affinity DataEC50:  2.70E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524899BDBM50524899(CHEMBL4458012)
Affinity DataEC50:  2.80E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524917BDBM50524917(CHEMBL4575028)
Affinity DataEC50:  2.90E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524949BDBM50524949(CHEMBL4445805)
Affinity DataEC50:  2.90E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524892BDBM50524892(CHEMBL4576878)
Affinity DataEC50:  3.00E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524887BDBM50524887(CHEMBL4446565)
Affinity DataEC50:  3.10E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in J-Lat 10.6 cells harboring LTR driven GFP reporter co-expressing CMV driven RFP reporter assessed as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524890BDBM50524890(CHEMBL4460170)
Affinity DataEC50:  3.10E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524875BDBM50524875(CHEMBL4439569)
Affinity DataEC50:  3.30E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524921BDBM50524921(CHEMBL4463494)
Affinity DataEC50:  3.60E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524882BDBM50524882(CHEMBL4465202)
Affinity DataEC50:  3.60E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524886BDBM50524886(CHEMBL4467303)
Affinity DataEC50:  3.70E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524879BDBM50524879(CHEMBL4531268)
Affinity DataEC50:  3.70E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524936BDBM50524936(CHEMBL4437444)
Affinity DataEC50:  4.30E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524957BDBM50524957(CHEMBL4445251)
Affinity DataEC50:  4.70E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524969BDBM50524969(CHEMBL4547664)
Affinity DataEC50:  4.70E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524960BDBM50524960(CHEMBL4522266)
Affinity DataEC50:  4.70E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524946BDBM50524946(CHEMBL4435131)
Affinity DataEC50:  4.70E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524958BDBM50524958(CHEMBL4559333)
Affinity DataEC50:  5.00E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50481920BDBM50481920(CHEMBL1075815)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of HIV1 TAT transfected to human HeLa cells assessed as decrease in luminescence after 48 hrs by duel luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524951BDBM50524951(CHEMBL4532989)
Affinity DataEC50:  6.30E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524916BDBM50524916(CHEMBL4439266)
Affinity DataEC50:  6.40E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524924BDBM50524924(CHEMBL4528111)
Affinity DataEC50:  6.40E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524884BDBM50524884(CHEMBL1386792)
Affinity DataEC50:  6.70E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50481917BDBM50481917(CHEMBL1075830)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of HIV1 TAT transfected to human HeLa cells assessed as decrease in luminescence after 48 hrs by duel luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50410417BDBM50410417(CHEMBL371627)
Affinity DataKd:  7.70E+3nMT: 2°CAssay Description:In vitro binding affinity towards Tat/TAR to determine interaction between TAR RNA and Tat peptide at room temperature using fluorescence spectrophot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524905BDBM50524905(CHEMBL4546726)
Affinity DataEC50:  8.00E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210164BDBM50210164(CHEMBL2132936)
Affinity DataEC50:  8.10E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in J-Lat 10.6 cells harboring LTR driven GFP reporter co-expressing CMV driven RFP reporter assessed as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524938BDBM50524938(CHEMBL4441342)
Affinity DataEC50:  9.20E+3nMAssay Description:Activation of Tat-mediated HIV1 transcription in HEK293- FlpIn-FM cells harboring LTR driven CBR reporter co-expressing CMV driven CBG reporter asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524888BDBM50524888(CHEMBL4540359)
Affinity DataEC50:  1.00E+4nMAssay Description:Activation of Tat-mediated HIV1 transcription in J-Lat 10.6 cells harboring LTR driven GFP reporter co-expressing CMV driven RFP reporter assessed as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
The Walter and Eliza Hall Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50398244BDBM50398244(CHEMBL609728)
Affinity DataEC50:  1.00E+4nMAssay Description:Inhibition of Tat-mediated transcription of viral promoter in 293 T cells transfected with HIV1 tat by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
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