Compile Data Set for Download or QSAR
Report error Found 50 of affinity data for UniProtKB/TrEMBL: P0A9A6
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203126BDBM50203126(Berberinechloride | 9,10-Dimethoxy-5,6-dihydro-[1,...)
Affinity DataKd:  23nMAssay Description:Displacement of bis-ANS from Escherichia coli FtsZMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 25525BDBM25525(CHEMBL490129 | 24-methyl-5,7,18,20-tetraoxa-24-aza...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of Escherichia coli recombinant FTsZ incubated for 10 mins in presence of GTP by spectrofluorimeter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399003BDBM50399003(CHEMBL2180486)
Affinity DataKd:  3.80E+3nMAssay Description:Binding affinity to Escherichia coli FtsZ at 25 degC by fluorescence anisotropy assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203065BDBM50203065(3-phenylprop-2-enal | cinnamaldehyde | 3-phenylacr...)
Affinity DataIC50: 5.81E+3nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203065BDBM50203065(3-phenylprop-2-enal | cinnamaldehyde | 3-phenylacr...)
Affinity DataIC50: 6.86E+3nMAssay Description:Inhibition of Escherichia coli FtsZ polymerizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079361BDBM50079361(CHEMBL3416824)
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086108BDBM50086108(CHEMBL3425702)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50439495BDBM50439495(CHEMBL2418095)
Affinity DataIC50: 9.87E+3nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203126BDBM50203126(Berberinechloride | 9,10-Dimethoxy-5,6-dihydro-[1,...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant Escherichia coli K12 FtsZ assembly by light-scattering assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079359BDBM50079359(Viriditoxin)
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 67454BDBM67454(MLS002473304 | purpurin | 1,2,4-tris(oxidanyl)anth...)
Affinity DataKd:  1.10E+4nMAssay Description:Binding affinity to Escherichia coli BL21 FtsZ assessed as dissociation constant of hydrophobic probe ANS-FtsZ complex fluorescence quenching incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079358BDBM50079358(CHEMBL3416948)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of Escherichia coli FtsZMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079359BDBM50079359(Viriditoxin)
Affinity DataIC50: 1.23E+4nMAssay Description:Inhibition of Escherichia coli FtsZ polymerizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079360BDBM50079360(CHEBI:69681 | Dichamanetin)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 25525BDBM25525(CHEMBL490129 | 24-methyl-5,7,18,20-tetraoxa-24-aza...)
Affinity DataIC50: 1.38E+4nMAssay Description:Inhibition of FtsZ in Escherichia coli assessed as disruption of Z ring formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086088BDBM50086088(CHEMBL3425706)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203126BDBM50203126(Berberinechloride | 9,10-Dimethoxy-5,6-dihydro-[1,...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of recombinant Escherichia coli K12 FtsZ GTPase activity by malachite green sodium molybdate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2018
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010058BDBM50010058(CHEBI:51231 | DAPI)
Affinity DataKd:  1.66E+4nMAssay Description:Binding affinity to Escherichia coli FtsZ by fluorescence anisotrophyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086098BDBM50086098(CHEMBL3425705)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086206BDBM50086206(CHEMBL3425606)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086123BDBM50086123(CHEMBL3425694)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086124BDBM50086124(CHEMBL3425693)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086201BDBM50086201(CHEMBL3425611)
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086200BDBM50086200(CHEMBL3425612)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086203BDBM50086203(CHEMBL3425609)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50439496BDBM50439496(CHEMBL2418096 | US9169182, J23)
Affinity DataIC50: 3.60E+4nMpH: 6.5 T: 2°CAssay Description:GTPase assays were performed in 50 mM MES, pH 6.5, 50 mM KCl, 5 mM MgCl2 in the presence of 2 uM FtsZ in the presence of varying concentrations of co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2016
Entry Details
US Patent

TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50439496BDBM50439496(CHEMBL2418096 | US9169182, J23)
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086197BDBM50086197(CHEMBL3425615)
Affinity DataIC50: 4.90E+4nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086109BDBM50086109(CHEMBL3425701)
Affinity DataIC50: 5.20E+4nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086199BDBM50086199(CHEMBL3425613)
Affinity DataIC50: 5.80E+4nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086120BDBM50086120(CHEMBL3425697)
Affinity DataIC50: 6.50E+4nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086105BDBM50086105(CHEMBL3425704)
Affinity DataIC50: 8.50E+4nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083355BDBM50083355(CHEMBL3423282)
Affinity DataIC50: 9.05E+4nMAssay Description:Inhibition of Escherichia coli ATCC 25922 recombinant N-His6-tagged FtsZ polymerization expressed in Escherichia coli BL21(DE3) incubated for 15 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086202BDBM50086202(CHEMBL3425610)
Affinity DataIC50: 9.50E+4nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086204BDBM50086204(CHEMBL3425608)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086107BDBM50086107(CHEMBL3425703)
Affinity DataIC50: 1.28E+5nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086116BDBM50086116(CHEMBL3425700)
Affinity DataIC50: 1.28E+5nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086118BDBM50086118(CHEMBL3425699)
Affinity DataIC50: 1.28E+5nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086119BDBM50086119(CHEMBL3425698)
Affinity DataIC50: 1.28E+5nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086121BDBM50086121(CHEMBL3425696)
Affinity DataIC50: 1.28E+5nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086122BDBM50086122(CHEMBL3425695)
Affinity DataIC50: 1.28E+5nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086125BDBM50086125(CHEMBL3425692)
Affinity DataIC50: 1.28E+5nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086180BDBM50086180(CHEMBL3425691)
Affinity DataIC50: 1.28E+5nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086191BDBM50086191(CHEMBL3425690)
Affinity DataIC50: 1.28E+5nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086196BDBM50086196(CHEMBL3425689)
Affinity DataIC50: 1.28E+5nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086198BDBM50086198(CHEMBL3425614)
Affinity DataIC50: 1.28E+5nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086205BDBM50086205(CHEMBL3425607)
Affinity DataIC50: 1.28E+5nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086207BDBM50086207(CHEMBL3425605)
Affinity DataIC50: 1.28E+5nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50086208BDBM50086208(CHEMBL3425604)
Affinity DataIC50: 1.28E+5nMAssay Description:Inhibition of Escherichia coli FtsZ GTPase activity after 5 mins by enzyme-coupled inhibition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2016
Entry Details Article
PubMed
TargetCell division protein FtsZ(Escherichia coli (strain K12))
University of Wisconsin-Madison

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 186046BDBM186046(US9169182, J24)
Affinity DataIC50: 1.60E+5nMpH: 6.5 T: 2°CAssay Description:GTPase assays were performed in 50 mM MES, pH 6.5, 50 mM KCl, 5 mM MgCl2 in the presence of 2 uM FtsZ in the presence of varying concentrations of co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2016
Entry Details
US Patent