Affinity DataIC50: 0.0200nMAssay Description:Inhibition of MMP8 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diaminopropionyl)Ala-Arg-NH2 as substrate incuba...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0300nMAssay Description:Inhibition of MMP8 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diaminopropionyl)Ala-Arg-NH2 as substrate incuba...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0400nMAssay Description:Inhibition of MMP8 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diaminopropionyl)Ala-Arg-NH2 as substrate incuba...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0460nMAssay Description:Inhibition of human recombinant MMP8More data for this Ligand-Target Pair
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of MMP-8 (unknown origin) using 7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 a...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0970nMAssay Description:Inhibition of human recombinant MMP8 using fluorescence peptide Cy3-PLGLK(Cy5Q)AR-NH2 substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0970nMAssay Description:Inhibition of human recombinant MMP8 using Cy3-PLGLK(Cy5Q)AR-NH2 as substrate after 40 mins by spectrofluorimetryMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0970nMAssay Description:Inhibition of recombinant human AMPA-activated MMP8 using Cy3-PLGLK(Cy5Q)AR-NH2 as substrate measured after 40 mins by spectrofluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0970nMAssay Description:Inhibition of APMA-activated recombinant human MMP-8 using Cy3-PLGLK(Cy5Q)AR-NH2 peptide as substrate measured after 40 mins by spectrofluorimetric m...More data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Initial rates of 4-nitrophenyl acetate hydrolysis catalyzed by different CA isozymes were monitored spectrophotometrically at 400 nm. A molar absorpt...More data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:The compound was tested for its binding affinity towards neutrophil collagenase (Matrix metalloprotease-8)More data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Inhibitory activity against the Matrix Metalloprotease-8More data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:The compound was tested for its binding affinity towards neutrophil collagenase (Matrix metalloprotease-8)More data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Inhibition of MMP8 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diaminopropionyl)Ala-Arg-NH2 as substrate incuba...More data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Inhibition of MMP-8 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:The compound was tested for its binding affinity towards neutrophil collagenase (Matrix metalloprotease-8)More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of MMP-8 (unknown origin) using 7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 a...More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of MMP-8 (matrix metalloprotease-8)More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of MMP-8 (unknown origin) using 7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 a...More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of MMP8 using (7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diaminopropionyl)Ala-Arg-NH2 as substrate incuba...More data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:The compound was tested for its binding affinity towards neutrophil collagenase (Matrix metalloprotease-8)More data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:The compound was tested for its binding affinity towards neutrophil collagenase (Matrix metalloprotease-8)More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of MMP-8 (unknown origin) using 7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 a...More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Initial rates of 4-nitrophenyl acetate hydrolysis catalyzed by different CA isozymes were monitored spectrophotometrically at 400 nm. A molar absorpt...More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of MMP-8 (unknown origin) using 7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 a...More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:The compound was tested for its binding affinity towards neutrophil collagenase (Matrix metalloprotease-8)More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:The compound was tested for its binding affinity towards neutrophil collagenase (Matrix metalloprotease-8)More data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:The compound was tested for its binding affinity towards neutrophil collagenase (Matrix metalloprotease-8)More data for this Ligand-Target Pair
Affinity DataKi: 0.340nMAssay Description:The compound was tested for its binding affinity towards neutrophil collagenase (Matrix metalloprotease-8)More data for this Ligand-Target Pair
Affinity DataKi: 0.350nMAssay Description:The compound was tested for its binding affinity towards neutrophil collagenase (Matrix metalloprotease-8)More data for this Ligand-Target Pair
Affinity DataKi: 0.390nMAssay Description:The compound was tested for its binding affinity towards neutrophil collagenase (Matrix metalloprotease-8)More data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of MMP-8 (unknown origin) using 7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 a...More data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human MMP8 assessed as cleavage of fluorogenic peptide MCAPro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human MMP8 assessed as cleavage of fluorogenic peptide MCAPro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of MMP-8 (unknown origin) using 7-methoxycoumarin-4-yl)acetyl-Pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl)Ala-Arg-NH2 a...More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibitors were assayed against purified hMMP-1, hMMP-2, hMMP-3, hMMP-8, hMMP-9, and hMMP-13 using an enzyme assay based on cleavage of the quenched ...More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibition of human Matrix metalloprotease-8More data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human MMP8 assessed as cleavage of fluorogenic peptide MCAPro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of matrix metalloprotease-8More data for this Ligand-Target Pair
Affinity DataKi: 0.410nMAssay Description:The compound was tested for its binding affinity towards neutrophil collagenase (Matrix metalloprotease-8)More data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:The compound was tested for its binding affinity towards neutrophil collagenase (Matrix metalloprotease-8)More data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:Inhibition of matrix metalloprotease-8More data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:The compound was tested for its binding affinity towards neutrophil collagenase (Matrix metalloprotease-8)More data for this Ligand-Target Pair
Affinity DataIC50: 0.470nMAssay Description:Inhibition of Matrix metalloprotease-8 (MMP-8) in fluorimetric assayMore data for this Ligand-Target Pair












































