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Report error Found 211 of affinity data for UniProtKB/TrEMBL: P82128
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50409669BDBM50409669(CHEMBL155514)
Affinity DataIC50: 0.457nMAssay Description:In vitro inhibition of porcine carboxylesterase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371969BDBM50371969(CHEMBL270374)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of pig liver carboxylesterase after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371971BDBM50371971(CHEMBL440542)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of pig liver carboxylesterase after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371969BDBM50371969(CHEMBL270374)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of pig liver carboxylesterase after 5 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371970BDBM50371970(CHEMBL89506)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of pig liver carboxylesterase after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371966BDBM50371966(CHEMBL269931)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of pig liver carboxylesterase after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371973BDBM50371973(CHEMBL402615)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of pig liver carboxylesterase after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50570553BDBM50570553(CHEMBL4854298)
Affinity DataIC50: 5nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50570555BDBM50570555(CHEMBL4868014)
Affinity DataIC50: 5.10nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371972BDBM50371972(CHEMBL270375)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of pig liver carboxylesterase after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371966BDBM50371966(CHEMBL269931)
Affinity DataIC50: 5.5nMAssay Description:Inhibition of pig liver carboxylesterase after 5 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371970BDBM50371970(CHEMBL89506)
Affinity DataIC50: 5.60nMAssay Description:Inhibition of pig liver carboxylesterase after 5 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50570549BDBM50570549(CHEMBL4853742)
Affinity DataIC50: 6.10nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50570554BDBM50570554(CHEMBL4858186)
Affinity DataIC50: 7.20nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50570551BDBM50570551(CHEMBL4853637)
Affinity DataIC50: 7.30nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50570550BDBM50570550(CHEMBL4849361)
Affinity DataIC50: 7.40nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371971BDBM50371971(CHEMBL440542)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of pig liver carboxylesterase after 5 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50570561BDBM50570561(CHEMBL4855838)
Affinity DataIC50: 7.70nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371971BDBM50371971(CHEMBL440542)
Affinity DataIC50: 8.32nMAssay Description:In vitro inhibition of porcine carboxylesterase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371968BDBM50371968(CHEMBL273138)
Affinity DataIC50: 8.60nMAssay Description:Inhibition of pig liver carboxylesterase after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371959BDBM50371959(CHEMBL86668)
Affinity DataIC50: 9.30nMAssay Description:Inhibition of pig liver carboxylesterase after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50409660BDBM50409660(CHEMBL155513)
Affinity DataIC50: 10.5nMAssay Description:In vitro inhibition of porcine carboxylesterase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371968BDBM50371968(CHEMBL273138)
Affinity DataIC50: 12nMAssay Description:Inhibition of pig liver carboxylesterase after 5 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371972BDBM50371972(CHEMBL270375)
Affinity DataIC50: 12nMAssay Description:Inhibition of pig liver carboxylesterase after 5 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50570552BDBM50570552(CHEMBL4855755)
Affinity DataIC50: 13nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50570559BDBM50570559(CHEMBL4868687)
Affinity DataKi:  14nMAssay Description:Competitive inhibition of porcine liver carboxylesterase by double reciprocal Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50409672BDBM50409672(CHEMBL153080)
Affinity DataIC50: 17.0nMAssay Description:In vitro inhibition of porcine carboxylesterase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371973BDBM50371973(CHEMBL402615)
Affinity DataIC50: 20nMAssay Description:Inhibition of pig liver carboxylesterase after 5 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371961BDBM50371961(CHEMBL270373)
Affinity DataIC50: 23nMAssay Description:Inhibition of pig liver carboxylesterase after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371959BDBM50371959(CHEMBL86668)
Affinity DataIC50: 25nMAssay Description:Inhibition of pig liver carboxylesterase after 5 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50570559BDBM50570559(CHEMBL4868687)
Affinity DataIC50: 28nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371965BDBM50371965(CHEMBL272075)
Affinity DataIC50: 28nMAssay Description:Inhibition of pig liver carboxylesterase after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371962BDBM50371962(CHEMBL155396)
Affinity DataIC50: 33nMAssay Description:Inhibition of pig liver carboxylesterase after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371970BDBM50371970(CHEMBL89506)
Affinity DataIC50: 37nMAssay Description:Inhibition of Sus scrofa (pig) carboxylesterase isolated from liver in using p-nitrophenyl acetate as substrate incubated for 5 min prior to substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371967BDBM50371967(CHEMBL257071)
Affinity DataIC50: 37nMAssay Description:Inhibition of pig liver carboxylesterase after 5 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50570556BDBM50570556(CHEMBL4847987)
Affinity DataIC50: 42nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50409670BDBM50409670(CHEMBL421992)
Affinity DataIC50: 43.6nMAssay Description:In vitro inhibition of porcine carboxylesterase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371967BDBM50371967(CHEMBL257071)
Affinity DataIC50: 46nMAssay Description:Inhibition of pig liver carboxylesterase after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50570560BDBM50570560(CHEMBL4872772)
Affinity DataIC50: 47nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50570557BDBM50570557(CHEMBL4856140)
Affinity DataIC50: 47nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50022772BDBM50022772(Isopropyl phosphorofluoridate | Neoglaucit | O,O'-...)
Affinity DataIC50: 50nMAssay Description:Inhibition of porcine liver carboxylesterase using [14C]GS-7340 substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371971BDBM50371971(CHEMBL440542)
Affinity DataIC50: 54nMAssay Description:Inhibition of Sus scrofa (pig) carboxylesterase isolated from liver in using p-nitrophenyl acetate as substrate incubated for 5 min prior to substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50570558BDBM50570558(CHEMBL4849436)
Affinity DataIC50: 56nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371965BDBM50371965(CHEMBL272075)
Affinity DataIC50: 63nMAssay Description:Inhibition of pig liver carboxylesterase after 5 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50529191BDBM50529191(CHEMBL4564380)
Affinity DataIC50: 70nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50412689BDBM50412689(CHEMBL460809)
Affinity DataIC50: 75nMAssay Description:Inhibition of Sus scrofa (pig) carboxylesterase isolated from liver in using p-nitrophenyl acetate as substrate incubated for 5 min prior to substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50570567BDBM50570567(CHEMBL4848799)
Affinity DataIC50: 89nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50371960BDBM50371960(CHEMBL155621)
Affinity DataIC50: 100nMAssay Description:Inhibition of pig liver carboxylesterase after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50570565BDBM50570565(CHEMBL4879228)
Affinity DataIC50: 102nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetLiver carboxylesterase(Pig)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50570566BDBM50570566(CHEMBL4849604)
Affinity DataIC50: 103nMAssay Description:Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
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