Compile Data Set for Download or QSAR
Report error Found 47 of affinity data for UniProtKB/TrEMBL: Q63704
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403039BDBM50403039(CHEMBL2216778)
Affinity DataIC50: 30nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403029BDBM50403029(CHEMBL2216792)
Affinity DataIC50: 40nMAssay Description:Inhibition of rat CPT1B expressed in intact Saccharomyces cerevisiae using [methyl-3H]carnitine by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403040BDBM50403040(CHEMBL2216779)
Affinity DataIC50: 55nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403037BDBM50403037(CHEMBL2216774)
Affinity DataIC50: 130nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403041BDBM50403041(CHEMBL2216776)
Affinity DataIC50: 150nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403038BDBM50403038(CHEMBL2216777)
Affinity DataIC50: 180nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50260111BDBM50260111(CHEBI:15531 | MALONYL-COENZYME A)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of rat heart mitochondrial CPT-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 80613BDBM80613(SMR000674573 | cid_9926449 | 1-(2,3,4-Trimethoxy-b...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of CPT1A in rat myocardiumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 80613BDBM80613(SMR000674573 | cid_9926449 | 1-(2,3,4-Trimethoxy-b...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of rat CPT1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50122839BDBM50122839([3-Carboxy-2-(3-tetradecyl-ureido)-propyl]-trimeth...)
Affinity DataIC50: 1.45E+3nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50101594BDBM50101594([3-Carboxy-2-(decane-1-sulfonylamino)-propyl]-trim...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50046145BDBM50046145(2-[6-hydroxy-4,4-dimethyl-6-pentadecyl-(2R,6S)-1,4...)
Affinity DataKi:  2.80E+3nMAssay Description:Compound was evaluated for its ability to inhibit carnitine palmitoyltransferase I activity in intact mitochondria from rat heartMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50101604BDBM50101604([3-Carboxy-2-(dodecane-1-sulfonylamino)-propyl]-tr...)
Affinity DataIC50: 3.40E+3nMAssay Description:In vitro inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50101598BDBM50101598([3-Carboxy-2-(dodecane-1-sulfonylamino)-propyl]-tr...)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50101589BDBM50101589([3-Carboxy-2-(nonylaminosulphonyl-amino)-propyl]-t...)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50101591BDBM50101591([3-Carboxy-2-(undecylaminosulphonyl-amino)-propyl]...)
Affinity DataIC50: 5.80E+3nMAssay Description:In vitro inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50101591BDBM50101591([3-Carboxy-2-(undecylaminosulphonyl-amino)-propyl]...)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50101600BDBM50101600([3-Carboxy-2-(undecylaminosulphonyl-amino)-propyl]...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50101600BDBM50101600([3-Carboxy-2-(undecylaminosulphonyl-amino)-propyl]...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50101598BDBM50101598([3-Carboxy-2-(dodecane-1-sulfonylamino)-propyl]-tr...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50101604BDBM50101604([3-Carboxy-2-(dodecane-1-sulfonylamino)-propyl]-tr...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50260115BDBM50260115(CHEMBL4097976)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of rat heart mitochondrial CPT-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 61402BDBM61402(perhexiline maleate | (Z)-but-2-enedioic acid;2-(2...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of rat heart mitochondrial CPT-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50260105BDBM50260105(CHEMBL1592481)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of Wistar rat heart mitochondrial CPT-1 assessed as reduction in conversion of palmitoyl CoA and L-carnitine into palmitoylcarnitine prein...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50260109BDBM50260109(CHEMBL4077250)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of rat heart mitochondrial CPT-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403034BDBM50403034(CHEMBL2114397)
Affinity DataIC50: 2.73E+4nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50260108BDBM50260108(CHEMBL4082420)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of rat heart mitochondrial CPT-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50122839BDBM50122839([3-Carboxy-2-(3-tetradecyl-ureido)-propyl]-trimeth...)
Affinity DataIC50: 4.34E+4nMAssay Description:In vitro inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50260104BDBM50260104(CHEMBL4081530)
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of rat heart mitochondrial CPT-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50122827BDBM50122827([3-Carboxy-2-(3-nonyl-ureido)-propyl]-trimethyl-am...)
Affinity DataIC50: 4.62E+4nMAssay Description:In vitro inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50260105BDBM50260105(CHEMBL1592481)
Affinity DataIC50: 7.70E+4nMAssay Description:Inhibition of rat heart mitochondrial CPT-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50122833BDBM50122833((3-Carboxy-2-octyloxycarbonylamino-propyl)-trimeth...)
Affinity DataIC50: 8.01E+4nMAssay Description:In vitro inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50101590BDBM50101590([3-Carboxy-2-(3-nonyl-ureido)-propyl]-trimethyl-am...)
Affinity DataIC50: 8.32E+4nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50260112BDBM50260112(CHEMBL4068222)
Affinity DataIC50: 8.80E+4nMAssay Description:Inhibition of rat heart mitochondrial CPT-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037268BDBM50037268((3R)-3-hydroxy-4-(trimethylammonio)butanoate | (-)...)
Affinity DataKi:  1.00E+5nMAssay Description:Tested against neonatal rat cardiac myocyte carnitine palmitoyltransferase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50122828BDBM50122828([3-Carboxy-2-(3-undecyl-ureido)-propyl]-trimethyl-...)
Affinity DataIC50: 1.18E+5nMAssay Description:In vitro inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50122834BDBM50122834([3-Carboxy-2-(3-dodecyl-ureido)-propyl]-trimethyl-...)
Affinity DataIC50: 1.20E+5nMAssay Description:In vitro inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50122836BDBM50122836([3-Carboxy-2-(3-tetradecyl-ureido)-propyl]-trimeth...)
Affinity DataIC50: 1.67E+5nMAssay Description:In vitro inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50101593BDBM50101593((3-Carboxy-2-octyloxycarbonylamino-propyl)-trimeth...)
Affinity DataIC50: 2.11E+5nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50260113BDBM50260113(CHEMBL4059578)
Affinity DataIC50: 2.15E+5nMAssay Description:Inhibition of rat heart mitochondrial CPT-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50122835BDBM50122835([3-Carboxy-2-(3-nonyl-ureido)-propyl]-trimethyl-am...)
Affinity DataIC50: 3.00E+5nMAssay Description:In vitro inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50122837BDBM50122837([3-Carboxy-2-(3-heptyl-ureido)-propyl]-trimethyl-a...)
Affinity DataIC50: 3.00E+5nMAssay Description:In vitro inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50122829BDBM50122829((3-Carboxy-2-octyloxycarbonylamino-propyl)-trimeth...)
Affinity DataIC50: 3.00E+5nMAssay Description:In vitro inhibition of [14C]palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50260114BDBM50260114(CHEMBL4079982)
Affinity DataIC50: 4.75E+5nMAssay Description:Inhibition of rat heart mitochondrial CPT-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50260110BDBM50260110(CHEMBL4097557)
Affinity DataIC50: 7.15E+5nMAssay Description:Inhibition of rat heart mitochondrial CPT-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2020
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037262BDBM50037262((R)-3-Hydroxy-5,5-dimethyl-hexanoic acid anion)
Affinity DataKi:  1.40E+6nMAssay Description:Tested against neonatal rat cardiac myocyte carnitine palmitoyltransferase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rat)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037261BDBM50037261(3-Hydroxy-5,5-dimethyl-hexanoic acid anion)
Affinity DataKi:  3.60E+6nMAssay Description:Tested against neonatal rat cardiac myocyte carnitine palmitoyltransferase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed