Compile Data Set for Download or QSAR
Report error Found 38 for UniProtKB: Q8BUY9
LigandChemical structure of BindingDB Monomer ID 31423BDBM31423(ethylenediamine scaffold, 4)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 50327998BDBM50327998(N-(2-((4-cyano-2-fluorophenyl)((1-methyl-1H-imidaz...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50327997BDBM50327997(N-(2-((4-cyanophenyl)((1-methyl-1H-imidazol-5-yl)m...)
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 13314BDBM13314(N-benzyl-N-{2-[(4-cyanophenyl)[(1-methyl-1H-imidaz...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50327993BDBM50327993(1-methyl-1H-imidazole-4-sulfonic acid biphenyl-3-y...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50327994BDBM50327994(1-methyl-1H-imidazole-4-sulfonic acid {2-[(4-cyano...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 13311BDBM13311(1-Methyl-1H-imidazole-4-sulfonic Acid {2-[(4-Cyano...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 13318BDBM13318(N-(4-cyanobenzyl)-N-(2-{(4-cyanophenyl)[(1-methyl-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50327983BDBM50327983(1-methyl-1H-imidazole-4-sulfonic acid {2-[(4-cyano...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50327990BDBM50327990(1-methyl-1H-imidazole-4-sulfonic acid {2-[(4-cyano...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 13317BDBM13317(N1-(tert-butyl)-N2-(2-{(4-cyanophenyl)[(1-methyl-1...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50327978BDBM50327978(N-(2-((4-cyanophenyl)((1-methyl-1H-imidazol-5-yl)m...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50327974BDBM50327974(N-Benzyl,N-{2-[(4-Cyanophenyl)-(3-methyl-3H-imidaz...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50327972BDBM50327972(1-methyl-1H-imidazole-4-sulfonic Acid Benzyl-{2-[(...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50327976BDBM50327976(N-benzyl-N-(2-((4-cyanophenyl)((1-methyl-1H-imidaz...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50327975BDBM50327975(N-benzyl-N-(2-((4-cyanophenyl)((1-methyl-1H-imidaz...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50327986BDBM50327986(N-(2-((4-cyanophenyl)((1-methyl-1H-imidazol-5-yl)m...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50327988BDBM50327988(N-(2-((4-cyanophenyl)((1-methyl-1H-imidazol-5-yl)m...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 13316BDBM13316(N-{2-[(4-cyanophenyl)[(1-methyl-1H-imidazol-5-yl)m...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 13315BDBM13315(1-Methyl-1H-imidazole-4-sulfonic Acid {2-[(4-Cyano...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50327987BDBM50327987(N-(2-((4-cyanophenyl)((1-methyl-1H-imidazol-5-yl)m...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50327984BDBM50327984(N-(2-((4-cyanophenyl)((1-methyl-1H-imidazol-5-yl)m...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50327977BDBM50327977(N-benzyl-N-(2-((4-cyanophenyl)((1-methyl-1H-imidaz...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50327981BDBM50327981(1-methyl-1H-imidazole-4-sulfonic acid (2-bromoally...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50327995BDBM50327995(N-(2-((4-cyanophenyl)((1-methyl-1H-imidazol-5-yl)m...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50327973BDBM50327973(1-methyl-1H-imidazole-4-sulfonic acid benzyl-{2-[(...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50327989BDBM50327989(N-(2-((4-cyanophenyl)((1-methyl-1H-imidazol-5-yl)m...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 13313BDBM13313(N-Benzyl-N-{2-[(4-cyanophenyl)-(3-methyl-3H-imidaz...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50327992BDBM50327992(1-methyl-1H-imidazole-4-sulfonic acid (3-cyanobenz...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50327991BDBM50327991(1-methyl-1H-imidazole-4-sulfonic acid {2-[(4-cyano...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 13308BDBM13308(N-benzyl-N-{2-[(4-bromophenyl)[(1-methyl-1H-imidaz...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50327982BDBM50327982(1-methyl-1H-imidazole-4-sulfonic acid {2-[(4-cyano...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50327980BDBM50327980(1-methyl-1H-imidazole-4-sulfonic acid {2-[(4-cyano...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50327979BDBM50327979(1-methyl-1H-imidazole-4-sulfonic acid allyl-{2-[(4...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 13307BDBM13307(1-Methyl-1H-imidazole-4-sulfonic Acid Benzyl-{2-[(...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 50327996BDBM50327996(1-methyl-1H-imidazole-4-sulfonic acid {2-[(4-cyano...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50327985BDBM50327985(N-(2-((4-cyanophenyl)((1-methyl-1H-imidazol-5-yl)m...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50327999BDBM50327999(N-(2-((5-cyanopyridin-2-yl)((1-methyl-1H-imidazol-...)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of Rap1A geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed