Compile Data Set for Download or QSAR
Report error Found 123 of affinity data for UniProtKB/TrEMBL: Q9UEW8
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM130909(US8822500, Stauro- sporine | US9920060, Staurospor...)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human STK39 using myelin basic protein as substrate preincubated for 20 mins followed by [gamma-33P]-ATP addition and measured after 12...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 14.4nMAssay Description:Inhibition of human STK39 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 17.2nMAssay Description:Inhibition of human STK39 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50630232(CHEMBL5433617)
Affinity DataIC50: 35nMAssay Description:Inhibition of STLK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50560445(CHEMBL4792789)
Affinity DataIC50: 50nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50560439(CHEMBL4762099)
Affinity DataIC50: 110nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataKd:  130nMAssay Description:Binding constant for STK39 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataKd:  140nMAssay Description:Binding constant for STK39 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataKd:  140nMAssay Description:Binding affinity to STK39More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2011
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM482158(TAE684 | BDBM50242742)
Affinity DataKd:  150nMAssay Description:Binding constant for STK39 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50560448(CHEMBL4759888)
Affinity DataIC50: 240nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50560415(CHEMBL4797256)
Affinity DataIC50: 260nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM31095(5-[(Z)-(5-fluoranyl-2-oxidanylidene-1H-indol-3-yli...)
Affinity DataKd:  430nMAssay Description:Binding constant for STK39 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50026612(BIBF-1120 | Nintedanib | Vargatef | US10981896, Co...)
Affinity DataKd:  520nMAssay Description:Binding constant for STK39 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM25118(4-amino-5-fluoro-3-[6-(4-methylpiperazin-1-yl)-1H-...)
Affinity DataKd:  530nMAssay Description:Binding constant for STK39 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50560424(CHEMBL4751500)
Affinity DataIC50: 650nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50355496(CHEMBL1908397)
Affinity DataKd:  890nMAssay Description:Binding constant for STK39 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50560420(CHEMBL4759820)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50308060(CEP-701 | 16-hydroxy-16-(hydroxymethyl)-15-methyl-...)
Affinity DataKd:  1.10E+3nMAssay Description:Binding constant for STK39 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50560419(CHEMBL4753158)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50308060(CEP-701 | 16-hydroxy-16-(hydroxymethyl)-15-methyl-...)
Affinity DataKd:  1.10E+3nMAssay Description:Binding affinity to STK39More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2011
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50560417(CHEMBL4750439)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM311210(US10155760, Example 66 | (S)-methyl (5-((2-amino-2...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of STLK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50560428(CHEMBL4783530)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM31085(cid_11409972 | 1-[4-[(4-ethylpiperazin-1-yl)methyl...)
Affinity DataKd:  1.50E+3nMAssay Description:Binding constant for STK39 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50560430(CHEMBL4758154)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50332294(N-tert-butyl-3-(5-methyl-2-(4-(2-(pyrrolidin-1-yl)...)
Affinity DataKd:  1.60E+3nMAssay Description:Binding constant for STK39 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50560429(CHEMBL4747390)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50355501(RUXOLITINIB PHOSPHATE | INCB-018424 | RUXOLITINIB ...)
Affinity DataKd:  1.90E+3nMAssay Description:Binding constant for STK39 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50560421(CHEMBL4793138)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50560433(CHEMBL4744527)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50560437(CHEMBL4748104)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50560438(CHEMBL4795291)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50560432(CHEMBL4757952)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50560418(CHEMBL4748683)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50560426(CHEMBL4757062)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50560444(CHEMBL4796271)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50560422(CHEMBL4762871)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM4552(CHEMBL288441 | SKI-606 | 4-[(2,4-Dichloro-5-methox...)
Affinity DataKd:  3.70E+3nMAssay Description:Binding constant for STK39 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50560440(CHEMBL4783506)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50350105(CHEMBL1814047)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50560416(CHEMBL4641560)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50560425(CHEMBL4796688)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50560423(CHEMBL4793886)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50560427(CHEMBL4758811)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of SPAK (unknown origin) by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM13535(N-(4-isopropoxyphenyl)-4-[6-methoxy-7-(3-piperidin...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for STK39 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM25013(4-[2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[(3S...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for STK39 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM5445(N-{3-chloro-4-[(3-fluorophenyl)methoxy]phenyl}-6-(...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for STK39 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM13336(4-{4-(4-fluorophenyl)-2-[4-(methylsulfinyl)phenyl]...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for STK39 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Human)
Center for Lymphoid Malignancies

Curated by ChEMBL
LigandPNGBDBM50326053(PKC-412 | CHEMBL608533 | US20240132489, Compound S...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to STK39More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2011
Entry Details Article
PubMed
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